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4-[(4-methoxyphenyl)methyl]-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-6-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-3-(quinolin-6-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
1-{2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
(3S,4S)-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
2-chloro-N-({1-[3-(methylsulfanyl)propanoyl]piperidin-3-yl}methyl)benzamide
2-[(4-methoxyphenyl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl (2S,4R)-1-[3-(azocan-1-yl)propanoyl]-4-hydroxypyrrolidine-2-carboxylate
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(thiophen-2-yl)propan-1-one
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(carbamoylmethyl)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)piperidine-3-carboxamide
1-[2-(propan-2-yloxy)phenyl]-3-[(3R)-pyrrolidin-3-yl]urea
methyl 4-(4-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-[2-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
2-[7-(hydroxymethyl)-9-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-ol
3-{4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazol-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-cyclopropyl-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]butanamide
(5S,9aS,9bS)-5-(1H-indol-3-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(1,3-benzoxazol-2-yl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]acetamide
1-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(3R,4R)-4-cyclopropyl-4-hydroxy-3-methyl-N-[(4-methylphenyl)methyl]piperidine-1-carboxamide
methyl 1-methyl-5-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]carbamoyl}-1H-pyrazole-3-carboxylate
3-methoxy-N-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
1-benzyl-6-hydroxy-4-[(5-methylfuran-2-yl)methyl]-1,4-diazepan-2-one
5-(2-fluorophenoxymethyl)-N-(2-phenylpropyl)-1H-pyrazole-3-carboxamide
2,4-dimethyl-N-(1-{4-[4-(pyrazin-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)benzamide
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[3-(4-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
ethyl 6-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
1-methyl-4-(4-propylpyrimidine-5-carbonyl)piperazine-2-carboxylic acid
8-{2-[(pyridin-2-ylmethyl)amino]benzoyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(2-phenylethyl)piperidine-1-carboxamide
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-{1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
3-[(3,4-dimethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-[3-amino-3-(3,4-dimethoxyphenyl)propanoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(2E)-N-[2-(4-methoxyphenyl)ethyl]-4-methyl-N-[(1-methylpiperidin-4-yl)methyl]pent-2-enamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
2-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-6-ethoxyphenol
[(1,5-dimethyl-1H-indazol-3-yl)methyl](1-phenoxypropan-2-yl)amine
methyl (2S,4S)-1-[(2,4-dimethylphenyl)methyl]-4-acetamidopyrrolidine-2-carboxylate
ethyl 4-[3-(1-methyl-1H-pyrazol-5-yl)propanamido]piperidine-1-carboxylate
9-[(2S)-2-hydroxy-2-phenylacetyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]urea
1-{4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-phenylpiperidin-1-yl)acetamide