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2-{4-[3-(1H-imidazol-2-yl)benzoyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
N-{1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}-N-methylacetamide
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl (2S)-2-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-2-phenylacetate
1-(2-{[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-3-ol
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
(2S,4S)-4-benzamido-1-cyclobutanecarbonyl-N,N-diethylpyrrolidine-2-carboxamide
4-[4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-6-methylpyrimidin-2-amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
N,N-dimethyl-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-2-carbonitrile
4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,2-dihydroquinazolin-2-one
(1s,4s)-4-hydroxy-N-{[4-(phenoxymethyl)thiophen-2-yl]methyl}cyclohexane-1-carboxamide
4-oxo-N-(1-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-4-phenylbutanamide
1-{[3-cyclopentyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(morpholine-4-carbonyl)pyridin-4-yl]azepane
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(4-phenoxybenzoyl)piperidine
2,7,8-trimethyl-4-(3-phenoxyazetidine-1-carbonyl)quinoline
N-(dicyclopropylmethyl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-9-methoxy-10-(4-methylpiperazine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
5-[4-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
(3aR,6aR)-2-cyclopropanecarbonyl-5-(4-methoxypyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopropyl-9-[2-(3-ethoxyphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-(2-fluoro-5-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
4-[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
N-({7-[4-(4-fluorophenyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
2-benzyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[(2-methoxyphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,5-dimethoxybenzamide
4-(4,6-dimethylpyridine-3-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(trifluoromethyl)pyridine
1-{4-[(2-aminopyridin-3-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
3-[(1-methylpyrrolidin-3-yl)methyl]-1-(2-phenoxyphenyl)urea
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-{4-[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]piperazin-1-yl}ethan-1-one
(3R,5S)-5-(morpholine-4-carbonyl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidine-3-carboxamide
(1S,5R)-6-(morpholine-4-sulfonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
{[(1R,5S,6S)-3-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(4-chlorophenyl)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-3-phenylpropanamide
5-(2,6-difluorophenoxymethyl)-N-[2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
6-(propan-2-yl)-N4-[3-(pyridin-3-yloxy)propyl]pyrimidine-2,4-diamine
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
2-methoxy-1-{4-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
3-({3-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}methyl)pyridin-2-amine
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione