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3-(piperidine-1-carbonyl)-1-propyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-fluoropyridine-2-carbonyl)pyrrolidin-3-yl]methanol
methyl 1-({[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]carbamoyl}methyl)-1H-pyrazole-3-carboxylate
methyl 3-[2-(4-fluorophenyl)acetyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
(4aR,7aS)-1-(2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-1-(2-butoxyacetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1R,3S)-3-methoxy-7-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-(3-methoxyphenyl)ethan-1-one
8-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
N-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanesulfonamide
2-chloro-4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-6-methoxyphenol
1-(3-chlorophenyl)-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
(1S,6R)-9-(9H-fluorene-9-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
5-butyl-4-(2-methoxyacetyl)-1-(2-methoxyphenyl)piperazin-2-one
N,6-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[(2,6-difluorophenyl)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(4-acetylphenyl)phenoxy]acetamide
6-[2-(azepan-1-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2S)-2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-3-phenylpropanamide
2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-methoxyethan-1-one
2-hydroxy-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-3,5-bis(propan-2-yl)benzamide
1-[2-(benzenesulfonyl)ethyl]-5-[4-(2-ethoxyphenyl)piperazin-1-yl]azepan-2-one
{4-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]morpholin-2-yl}methanamine
N-[3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]cyclobutanecarboxamide
N-(3-methoxypropyl)-1-methyl-5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-cyclopropyl-3-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
1-[1-(5-hydroxypyrazine-2-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(1R,3S)-7-(2-ethylpyridine-4-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
(1S,5R)-3-cyclobutanecarbonyl-6-(3,5-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethylamino)ethyl]-4-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
(1R,6S)-N-[2-(furan-2-ylmethoxy)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-methoxybenzoyl)piperidine
2-chloro-N-{[1-(pent-4-enoyl)piperidin-3-yl]methyl}benzamide
1-(2-{1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-{2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}-4-methyl-1,4-diazepane
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopent-1-ene-1-carboxamide
2-[5-(1,1-dioxo-1λ6-thian-4-yl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
methyl 2-(8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetate
3-amino-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
N-cyclopropyl-4-methoxy-2-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzamide
N-[4-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol