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(2R,6R)-4-[(5-ethylfuran-2-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane
N-[3-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)pyridin-2-yl]-2,2-dimethylpropanamide
4-methoxy-N-{[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-(1-benzofuran-2-ylmethyl)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1,5,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({8-[(2,4-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
3-(3,4-difluorophenyl)-5-[5-(methoxymethyl)furan-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-(3-{[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-2-methyl-1,4-dihydropyridin-4-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyrazin-2-amine
1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
ethyl 1-benzyl-5-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(carbamoylmethyl)-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamide
2-amino-4-(2,4-dimethoxy-3-methylphenyl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
2-[5-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)furan-2-yl]benzonitrile
9-(1-benzylpyrrolidine-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
5-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)-2-(pyrrolidin-1-yl)pyrimidine
5-[(3-chloro-4,5-dimethoxyphenyl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[4-(thiophen-2-yl)-1H-imidazol-1-yl]pyridine-3-carboxamide
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-[4-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R)-2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
4-benzyl-3-ethyl-1-(3-methyl-1,2-oxazole-5-carbonyl)-1,4-diazepan-5-one
4-benzyl-1-(2-cyclopropylpyrimidine-5-carbonyl)-3-ethyl-1,4-diazepan-5-one
(1,3-benzothiazol-2-ylmethyl)({[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3,5-dihydroxy-4-methyl-N-(3-phenylprop-2-yn-1-yl)-N-propylbenzamide
1-(methoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)cyclobutane-1-carboxamide
5-chloro-2-methoxy-4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenol
4-(1-{4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]phenyl}ethyl)morpholine
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-(cyclopropylmethyl)-1-methyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[3-(1H-pyrazol-1-yl)propyl]amine
4-(1H-pyrazol-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
methyl 3-(2-cyclohexylacetyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl (2S,4R)-4-(quinoline-2-amido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl)pyridine
N-(4-chlorophenyl)-3-(3,4-dimethoxybenzoyl)piperidine-1-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
6-ethyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
2-(1-benzyl-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-2-yl)ethan-1-ol
3-methyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyridazine
5-{1-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
[(5-fluoro-1H-indol-2-yl)methyl]({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)methylamine
3-(pyridin-4-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
N-(3-methoxyphenyl)-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}propanamide
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yl)ethyl]benzamide
N-(1-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-amino-6-(4-hydroxyphenyl)-5-methyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile