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6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-2-one
[2-({4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one
7-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
2-({2-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{3-[2-(benzyloxy)ethyl]-4-fluorophenyl}ethan-1-one
4-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carbonyl}morpholine
(2S)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
(2S)-N2-ethyl-N1-[3-(2-methoxyphenyl)phenyl]pyrrolidine-1,2-dicarboxamide
N-({2-[3-(piperidine-1-carbonyl)phenyl]phenyl}methyl)propanamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(dicyclopropylmethyl)methylamine
4-(cyclohexylmethyl)-1-[(2E)-2-methylbut-2-en-1-yl]-1,4-diazepan-5-one
N-[6-(phenylamino)pyridin-3-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-N-ethyl-4-{4-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
[1-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
(1S,5R)-6-(cyclopropylmethyl)-3-(3,5-dimethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-3-methyl-1,2-oxazole
methyl 4-{[2-(3-methoxyphenyl)-1,3-benzoxazol-6-yl]formamido}butanoate
8-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
N-(1-{7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-4-methoxybenzamide
2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
7-[(2-fluorophenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
2,6-dimethyl-N-({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)pyrimidine-4-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
methyl[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](naphthalen-1-ylmethyl)amine
N-{[8-(1,3-benzothiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}oxane-4-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(1-methoxypropan-2-yl)piperidine-3-carboxamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)azepane-1-sulfonamide
4-(1-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}cyclohexyl)morpholine
N-cyclopentyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-methoxy-N-{[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-ethyl-N,N-dimethyl-3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-amine
4-[10-(methoxycarbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-3-carbonyl]pyridin-1-ium-1-olate
N,3,5,7-tetramethyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
6-(benzyloxy)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methylphenoxy)ethan-1-one
N-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}methanesulfonamide
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenol
1-methyl-4-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazine
methyl 6-[(2-methylpiperidin-1-yl)methyl]-3-(thiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]piperidine-4-carboxamide
1-[2-(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-[1-(3-phenyl-1,2-oxazole-5-carbonyl)azetidin-3-yl]pyridine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(trifluoromethyl)pyrimidin-4-amine
3-[(3,4-difluorophenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S)-2-amino-1-(3,3-diphenylpiperidin-1-yl)-3-(1H-imidazol-4-yl)propan-1-one