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{1-[(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidin-2-yl}methanol
N-[(1R)-1-(4-methoxyphenyl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)[2-(2-methoxy-4-methylphenoxy)ethyl]amine
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
5-(3-cyclohexylpropyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-amino-3-ethyl-N-[2-(pyridin-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{3-[4-(6-chloropyridazin-3-yl)piperazin-1-yl]-2,2-dimethylpropyl}morpholine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
(4aR,8aS)-6-[(4-methylphenyl)methyl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-amine
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
(3R,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-cyclopropyl-N,N-dimethylpyrrolidin-3-amine
5-acetamido-N-[2-(4-fluorophenyl)ethyl]-1-(2-methoxyethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-4-methyl-1H-imidazole
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2,3-dimethylquinoxalin-6-yl)-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
8-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[3-(pyridin-4-yl)azetidin-1-yl]pyridine-3-carboxylic acid
3-(2-fluorophenyl)-1-methyl-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-2,5-dione
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
6-methyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-[2-(1H-indazol-3-yl)acetyl]pyrrolidine-2-carboxylate
dimethyl[3-(2-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
N-benzyl-3-({[(5-ethylpyridin-2-yl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-cyclopentyl-4-{1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carbonyl}piperazin-2-one
N,3,4,7-tetramethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-4-(morpholin-4-yl)benzamide
(2-{2-[1-(4-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(oxan-2-ylmethyl)propanamide
1-(oxan-4-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
7-(3,4-dimethoxyphenyl)-4-[(2-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
{3-ethyl-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}methanol
5-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)-1H-1,2,3,4-tetrazole
1-[2-(diethylamino)ethyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
N-{[3-methyl-7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}methanesulfonamide
2-methanesulfonamido-N-[(3R,4S)-4-propyl-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]acetamide
methyl 1-(2-methoxyethyl)-5-[(3-methylbutyl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 2-{1-[(2-hydroxy-3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetate
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-ethyl-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
2-cyclopentyl-9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({3-[3-(pyridin-4-yl)propoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)naphthalene-1-sulfonamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
methyl (2S)-2-{[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}-3-methylbutanoate
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)propanamide
N-{[3-methyl-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}propanamide
1-{[(cyclohexylmethyl)carbamoyl]methyl}-3-(3-methoxypropyl)piperidine-3-carboxylic acid
ethyl 1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate