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(2R,4R)-4-hydroxy-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}pyrrolidine-2-carboxamide
methyl (2R,4S)-4-hydroxy-1-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}piperidine-2-carboxylate
2-[4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
1-(2-methoxyacetyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
4-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]-2,6-dimethylpyrimidine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
N,N-bis(propan-2-yl)-2-(1-propyl-1H-1,2,4-triazol-5-yl)benzamide
5,6-dimethyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]thieno[2,3-d]pyrimidine
N-{2-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}-2-methylpropanamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
2-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(furan-2-carbonyl)-1,4-diazepane
5-(methanesulfonylmethyl)-2-[3-(1H-pyrazol-5-yl)phenyl]pyridine
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-{[4-(morpholin-4-yl)phenyl]methyl}propanamide
2-(2-methyl-1H-indol-3-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(6-cyanopyridin-3-yl)-1-[3-(morpholin-4-yl)propyl]urea
2-(2-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenoxy)acetic acid
N-(2-hydroxyethyl)-2-(trimethyl-1H-pyrazol-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
(3aR,7aS)-2-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
5-[1-(2,2-diphenylethyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
5-(3-fluoro-4-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl 4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
N-benzyl-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
6-methyl-3-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,N-dimethylpyrazin-2-amine
7-(cyclobutylmethyl)-2-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(1S,6R)-9-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
1-({1-[1-(ethanesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
1-{4-fluoro-2-[3-(1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-one
2-chloro-N-ethyl-N-(oxolan-2-ylmethyl)-5-(1H-pyrazol-1-yl)benzamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[1-(1,3-thiazol-2-yl)propyl]urea
1-[1-(1-ethylpiperidin-4-yl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
3-[2-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-2-oxoethyl]-1,2,3-oxadiazol-3-ium-5-olate
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
(1S,5R)-3-methyl-6-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[4-(piperidin-1-yl)piperidin-1-yl]methyl}-4-(pyridin-3-yl)phenol
ethyl 3-[(2-methylphenyl)methyl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylate
N-[1-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-decahydro-1,6-naphthyridin-2-one
8-{5-[ethyl(methyl)carbamoyl]pyridin-2-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]methyl}pyrimidin-2-amine
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-cyclopentyl-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepane
N-[2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4,6-dimethoxy-1,3,5-triazine