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1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazine
N-cyclobutyl-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
4-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carbonyl)morpholine
4-(3,6-dimethylpyrazin-2-yl)-2-(2-phenylethyl)morpholine
(2E)-3-(2-fluorophenyl)-N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)prop-2-enamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-[(4-fluorophenyl)formamido]-N-methylpropanamide
1-{4-[(oxan-2-ylmethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-(3-phenylpropyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(thiophen-2-yl)ethyl]acetamide
N-[4-(3-fluorophenyl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-3-carboxamide
N-({7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
2,5-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}quinoxaline
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-(pyridin-3-ylmethyl)piperidin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-5-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(2-methoxyphenyl)-4-[(3E)-pent-3-enoyl]piperazin-2-one
3-acetyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1-(azepan-1-yl)-3-(2-methoxy-4-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidine-4-carboxylate
[(3R,4R)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2,7,8-trimethyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoline
2-{5-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-[(3R,4R)-3-hydroxy-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl]pyrazine-2-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(5-hydroxyadamantan-2-yl)propanamide
4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazole
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
6-methoxy-3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]quinoline
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-(1H-imidazol-2-yl)piperidine
2-(2-phenylethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
3-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]-3-methyl-1λ6-thiolane-1,1-dione
3-(methylsulfanyl)-N-{[8-(thiophene-2-sulfonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-amine
N-cyclopentyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
2-methoxy-1-{4-[2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-(butan-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}pyridine-2,4-diol
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-ethyl-3-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-[(3-methylphenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
1-{1'-[(2-chloro-4-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)azepane
[(2,6-dimethoxyphenyl)methyl](methyl)[(1-methylpiperidin-3-yl)methyl]amine
6-(4-methoxyphenyl)-3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propane-1,3-diol