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methyl 4-{4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}benzoate
(3R,4R)-1-(2,5-dimethylpyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-[(2-methoxy-3,5-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-amine
2-{4-[2-(3-cyano-2-methyl-1H-indol-1-yl)acetyl]morpholin-3-yl}-N-(2-fluoroethyl)acetamide
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
4-(4-chlorophenyl)-1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}butan-1-one
3-({[(3-chlorophenyl)methyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
1-[1-(butan-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-ethyl-1-[3-(pyrrolidine-1-carbonyl)benzenesulfonyl]-2,5-dihydro-1H-pyrrole
5-[2-(aminomethyl)piperidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]pyrimidin-4-ol
4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-methyl-8-(2-methylpropyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinoxaline
1-cyclopentyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-4-yl}-N-phenylpropanamide
1-[(2-chlorophenyl)methyl]-3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3,6-dimethylpyrazin-2-yl)piperidin-3-ol
N-cyclopropyl-1-{1-[1-(4-hydroxyphenyl)propan-2-yl]piperidin-4-yl}piperidine-4-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl]methanol
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-difluorobenzamide
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-cyclobutanecarbonyl-1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(5-hydroxyadamantan-2-yl)-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-(4-acetylphenyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-methylthiophene-2-carboxamide
N-(1-phenylcyclopropyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-cyclopropyl-1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]propan-1-one
N,N-dimethyl-5-(6-methylquinolin-5-yl)thiophene-2-carboxamide
2-fluoro-N-(1-{[(2-hydroxy-2-phenylethyl)(methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)benzamide
(2-{2-[3-(morpholin-4-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)urea
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
3-[1-(6-aminopyridin-2-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
2-(5-chloro-2-methoxyphenyl)-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]acetic acid
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
N-(3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-3-oxopropyl)acetamide
1-[(2-fluorophenyl)methoxy]-8-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
3-{5-[1-(3-chlorophenoxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-(butan-2-yl)-4-methoxy-N-(thiophen-3-ylmethyl)cyclohexane-1-carboxamide
(2E)-N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-methyl-3-propyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-5-carboxamide
[1-(2,7-dimethylquinoline-4-carbonyl)piperidin-4-yl](pyridin-3-yl)methanol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
methyl 1-[(3S,5S)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(2-methoxyethyl)-2-(1-methyl-1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(dimethylamino)ethyl]-1-[3-(3-fluorophenyl)phenyl]-3-(oxolan-2-ylmethyl)urea