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1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
methyl 3-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]propanoate
4-[2-(2,6-difluorophenyl)acetyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[4-(2-methoxyethyl)piperazin-1-yl]propan-1-one
methyl (2S,4R)-1-methyl-4-[3-(propan-2-yl)-1H-pyrazole-5-amido]pyrrolidine-2-carboxylate
2-{3-[3-(6-methoxypyridin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-(2-{4-[5-(4-methoxyphenyl)furan-2-carbonyl]piperazin-1-yl}ethoxy)ethan-1-ol
2-(2H-1,3-benzodioxole-5-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(cyclohexylmethyl)amino]-N-[(3S)-2-oxoazepan-3-yl]-5-[(propan-2-yl)sulfamoyl]benzamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-pyrazole-4-carboxamide
8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(2-methylphenyl)piperidine
[(2S,6S)-4-[4-(diethylamino)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-({7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(4-methanesulfonylphenyl)methyl]methylamine
1,7-dimethyl-2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
(2R,6R)-10-methoxy-4-[3-(methylsulfanyl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-{4-[3-(piperidin-3-yl)benzoyl]piperazin-1-yl}ethoxy)ethan-1-ol
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(5-chlorothiophen-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
{2-[2-(propan-2-yloxy)phenyl]quinolin-3-yl}methanol
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-[4-(1-benzofuran-5-ylmethyl)morpholin-3-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
(4aR,7aS)-1-ethyl-4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
4-methoxy-6-[4-(2-methoxybenzoyl)piperazin-1-yl]pyrimidin-2-amine
5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
5-methoxy-3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1H-indazole
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-{4-[6-(cyclopropylamino)pyridazin-3-yl]phenyl}propanoic acid
4-{4-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperazin-1-yl}-2-(2-methoxyethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(4-ethyl-5-methylthiophen-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{2-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]ethyl}-5-methyl-1,2,4-oxadiazole
N-[2-(2,4-difluorophenyl)-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-cycloheptyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
N-[4-(furan-2-yl)phenyl]-1-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]piperidine-3-carboxamide
1-(3-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
3-(4-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-1-yl)propanamide
N-[(3,4-difluorophenyl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-[(4-phenylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2R)-2-amino-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
1-methoxy-8-[3-(trifluoromethyl)benzoyl]-1,8-diazaspiro[4.5]decan-2-one
N-cycloheptyl-4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(4-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-phenylpropanamide
3-methyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole