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1-{2-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-4-ol
N-(2-methoxyethyl)-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
1-(1H-imidazol-4-ylmethyl)-4-(1H-indazole-3-carbonyl)-1,4-diazepan-6-ol
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(3-methyl-1H-pyrazol-5-yl)methyl]amine
3-(1,3-benzoxazol-2-ylmethyl)-6-ethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-({1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
1-(2-methylpropyl)-5-(1,2,3,6-tetrahydropyridin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1-(3-hydroxyphenyl)pyrrolidin-2-one
[(3S,5R)-1-(5-ethylthiophene-3-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-cyclopentyl-3-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-4-chloro-2-methylbenzamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-methyl-2-(pyrrolidin-1-yl)propan-1-one
1-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
(2S)-N2-benzyl-N2-[(3-methylpyridin-2-yl)methyl]pyrrolidine-1,2-dicarboxamide
methyl 3-[(3S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol
5-[4-(oxan-4-yl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-(piperidine-1-carbonyl)-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]pyrazine
4-{4-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperazin-1-yl}-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
5-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
ethyl 1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
2-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
N-(1,4-dioxan-2-ylmethyl)-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-[(2R)-1-hydroxypropan-2-yl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
N-[(4-methylphenyl)methyl]-1-[2-(2-methylpropanamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-ol
2-[(pyridin-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methylphenyl)acetamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
4-{1-benzyl-5-[3-(furan-2-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
{3-[5-(1-methyl-1H-imidazol-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
2,6-dimethyl-4-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}phenyl acetate
2-(propan-2-yl)-8-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]-N-(oxolan-2-ylmethyl)acetamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
2-(3-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
1-(adamantan-1-yl)-4-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}piperazine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyrrolidin-2-one
(3S,9aR)-3-(4-aminobutyl)-8-[(5-chlorothiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
7-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
2-methyl-4-[4-(1,4-oxazepan-4-ylmethyl)phenyl]butan-2-ol
ethyl 1-[5-(cycloheptylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carbonyl]piperidine-3-carboxylate
N'-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N'-(pyridin-3-ylmethyl)butanediamide