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N,N-diethyl-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
4-fluoro-N-[(1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]benzamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-ethyl-5-methoxy-N-(2-methylprop-2-en-1-yl)benzamide
[(3R,4R)-1-(3-fluoropyridin-2-yl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenoxyethan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(3-methoxyphenyl)acetamide
1-[(2-fluorophenyl)methyl]-4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazin-2-one
2-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
3-hydroxy-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
4-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
1-cycloheptyl-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
N-[1-(7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]-2-methoxyacetamide
N4-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-4,6-diamine
6-methoxy-3-methyl-N-[2-(1,3-thiazol-2-yl)ethyl]-1-benzofuran-2-carboxamide
methyl 9-[(4-fluorophenyl)methoxy]-3-[(3-hydroxy-4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2,2-dimethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
(3S,4S)-3-hydroxy-4-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)-1λ6-thiolane-1,1-dione
9-[(5-propylfuran-2-yl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 9-[(4-fluorophenyl)methoxy]-3-(2-methylpropyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(furan-3-ylmethyl)methylamine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
(2S)-2-amino-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
[(3aS,6aS)-2-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
propyl (4aR,7aS)-4-(2-methylpyrimidine-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-(naphthalen-1-ylmethyl)-4-{4-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
6-[3-(3-methyl-3-phenylpiperidin-1-yl)-3-oxopropyl]-2,3,4,5-tetrahydropyridazin-3-one
4,6-dimethyl-5-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-2H-pyran-2-one
1-[2-(furan-2-ylmethoxy)phenyl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
N-(3-hydroxypropyl)-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2S,4S)-4-amino-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{4-[3-(ethylsulfanyl)phenyl]-1H-pyrazol-1-yl}propanamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrimidine
N-(3-methyl-1-propyl-1H-pyrazol-5-yl)-3-[(2-methylpyrrolidin-1-yl)methyl]benzamide
N-(1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-2-[3-(3-fluorophenyl)-1H-pyrazol-1-yl]acetamide
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(piperidin-3-yl)benzamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-(3-methylbutyl)acetamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(1,3-thiazol-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 2-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoate
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2,5-dimethyl-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
(3aR,6aR)-2-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
2-amino-4-(4-cyanophenyl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide