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2-[4-(4-amino-5-methylpyrimidin-2-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-3-yl}pyrimidine
N-[(2R,3R)-2-methoxy-1'-[2-(phenylsulfanyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
methyl (2S)-1-({2-[4-(methoxycarbonyl)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)pyrrolidine-2-carboxylate
4-(4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)but-3-yn-1-ol
13-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-{1-[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
2-{4-[4-(ethylamino)pyrimidin-2-yl]piperazin-1-yl}-N-phenylacetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-(1-phenylbutyl)benzamide
1-(3-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
(3S,5R)-1-(2-phenylethyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
methyl 5-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[1-(4-fluorophenyl)propyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(azepane-1-sulfonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-[5-(methoxymethyl)thiophene-2-carbonyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)piperidin-2-one
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(5-fluoropyrimidin-2-yl)piperidine-4-carboxylic acid
3-{5-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[4-(6-methoxypyridazin-3-yl)phenyl]methanesulfonamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
4-(2-methylphenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
methyl 1-{[1-(dimethylcarbamoyl)ethyl]carbamoyl}cyclopropane-1-carboxylate
5-[(2-chloro-5-methoxy-4-propoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 1-ethyl-5-{[(5-methylthiophen-2-yl)methyl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}benzoic acid
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(1S,5R)-6-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-phenylethyl)-5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-benzoxazole
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-6-ethyl-2-methylquinoline-4-carboxamide
2-{1-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-(4-{4-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}phenyl)cyclopentanecarboxamide
4-(4-methoxyphenoxy)-1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
N-methyl-2-(methylamino)-N-phenyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
2-(2-phenylethyl)-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(1H-pyrazol-5-yl)phenyl]pyridine-4-carbonitrile
3-{2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}-4-methyl-1,2,5-oxadiazole
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
3-(3-methoxyphenyl)-N,N-bis(prop-2-en-1-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
2,3-dimethyl-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}quinoxaline-6-carboxamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]pyrrolidin-3-amine
7-(2-acetylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]pyridine
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-phenyl-1,2-oxazole-5-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
6-chloro-3-({[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
3-{[(diphenylmethyl)amino]methyl}-7-methoxy-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
1-(4-benzylpiperidin-1-yl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]propan-1-one
N-({5-methyl-2-[3-(5-methylthiophene-2-amido)phenyl]-1,3-oxazol-4-yl}methyl)quinoline-2-carboxamide
2-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]phenoxy}ethan-1-ol