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N-(5-oxo-1-phenylpyrrolidin-3-yl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
7-(3-chlorophenyl)-4-(2,3-dihydro-1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(1-methyl-1H-pyrazole-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(furan-2-ylmethyl)piperidine-3-carboxamide
5-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)furan-2-yl]benzonitrile
2-(4-{3-[(3-ethylphenyl)carbamoyl]propanoyl}morpholin-3-yl)acetic acid
2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-ol
1-{5-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-[2-(aminomethyl)morpholin-4-yl]-N-(2,4-dimethoxyphenyl)pyridine-3-carboxamide
1,4,6-trimethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-fluorophenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}cyclopropane-1-carboxamide
N-tert-butyl-7-[(4-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(3,3-dimethylbutyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-methyl-3-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
2-[3-({[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)phenoxy]acetamide
1-{[3-(3-methoxypiperidine-1-carbonyl)-1H-pyrazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-(cyclohexylmethyl)-N5-[2-(4-methoxyphenyl)ethyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(but-2-ynoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
1-[(3-methylphenyl)methyl]-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1H-indole
N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
(3R,5R)-5-(morpholine-4-carbonyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
(3S,4S)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3-phenyl-1H-pyrazole-4-carboxamide
(1s,4s)-N-[(4-methoxyphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
6-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine-2-carbonitrile
4-(2H-1,3-benzodioxol-5-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{2-[5-methyl-4-({2-[4-(methylsulfanyl)phenyl]acetamido}methyl)-1,3-oxazol-2-yl]phenyl}cyclobutanecarboxamide
2-[4-(3-methoxypropyl)piperazine-1-carbonyl]-3,5-dimethyl-1H-indole
1-[4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}sulfonyl)phenyl]ethan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N,2,5,6-tetramethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidin-4-amine
N-(2,3-dihydro-1H-inden-2-yl)-2-[(dimethylamino)methyl]-N-methyl-1,3-thiazole-4-carboxamide
1-(2-methoxy-2-methylpropyl)-2-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
3-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(furan-2-yl)propanamide
1-({5-[(2,6-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-[4-(morpholine-4-sulfonyl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
N-[(3R,4S)-1-[(2-chloro-4,6-dimethoxyphenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]acetamide
2-[1-(cyclopropylmethyl)-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-yl]ethan-1-ol
N-[2-(4-phenylpiperidin-1-yl)ethyl]morpholine-2-carboxamide
3-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea