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N-cyclopropyl-2,5-dimethoxy-N-{[3-(2-methylpropoxy)phenyl]methyl}benzamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3-ethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
4-{3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2,5-dimethyl-1H-pyrrol-1-yl}-4H-1,2,4-triazole
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-[1-(thiophen-2-yl)propyl]urea
3-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)butanamide
4-phenyl-6-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
4-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydrophthalazin-1-one
N-{[4-(difluoromethoxy)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
4-[5-(1-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazol-3-yl]pyridine
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-methyl-1,2,4-oxadiazole
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
2-acetyl-8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-methyl-1H-1,2,3-benzotriazole-4-sulfonamide
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
(1S,5R)-3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(cyclobutylsulfamoyl)-N-(1,4-dioxan-2-ylmethyl)-N-methylbenzamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
3-hydroxy-2-methyl-N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)benzamide
N-(1-{7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}thiophen-3-yl)prop-2-yn-1-ol
N-cycloheptyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propanamide
4-[(6-chloroquinolin-2-yl)methyl]morpholine-2-carboxamide
N-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
methyl 2-{methyl[(1-methylpiperidin-3-yl)methyl]carbamoyl}benzoate
3-methyl-N-[2-(4-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}phenoxy)ethyl]thiophene-2-carboxamide
2-cyclopentyl-8-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-methyl-3-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-(3-methoxyphenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
1,3-dimethyl-2,6-dioxo-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-methyl-2-(propan-2-yl)-N-[(4-sulfamoylphenyl)methyl]-1,3-thiazole-5-carboxamide
N-benzyl-5-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrimidin-2-amine
1-(4-methoxybenzoyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
N-[2-(pyridin-4-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(dimethylamino)-1-[(2R,3R)-2-hydroxy-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]ethan-1-one
1-[(2-fluorophenyl)methyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5,5-dimethyl-3-(4-phenoxybutyl)-1,3-oxazolidine-2,4-dione
N-[(2-methoxyphenyl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-[1-(1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
3-{[5-(1-ethylpiperidin-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
3-(aminomethyl)-4-(4-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-methyl-2-(4-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-[2-(methylsulfanyl)phenyl]acetic acid
1-(cyclohexylmethyl)-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide