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5-{3-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
8-(1-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-3-yloxy)acetamide
[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine
5-[(4-benzoylpiperazin-1-yl)methyl]-1H-indole
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}piperidin-2-one
(3S,4S)-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
2-{1-[1-(2,6-difluoro-3-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
5,6-dimethyl-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
2-(propan-2-yl)-5-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}pyrimidine
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
2-(2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)ethan-1-ol
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
8-(cyclopentylmethyl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrazine
8-cyclobutanecarbonyl-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}amino)-N-(2,4,6-trimethylphenyl)propanamide
2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-methylpropanamide
4-(pyridin-3-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]pyrimidin-2-amine
methyl 1-{9-methoxy-3-[(5-methylfuran-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
3-({[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl)amino}methyl)benzonitrile
(3aR,5S,6S,7aS)-2-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
4,5-dimethyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-2-(3-methoxyphenyl)pyrrolidine-1-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]propan-1-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(pyridin-4-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]propanamide
1-[(4-methoxyphenyl)methyl]-5-[3-(methylsulfanyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
8-methoxy-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
2-(3-{1,4-diazabicyclo[3.2.2]nonan-4-ylmethyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-(1,2-oxazol-3-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3-ethoxy-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
(7-methyl-2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}quinolin-3-yl)methanol
1-methyl-4-[(2-{[3-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)methyl]piperazine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(benzyloxy)butan-1-one
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-(cyclohex-1-en-1-yl)-1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
1-(3-chloro-2,6-dimethylphenyl)-3-[(2S)-pyrrolidin-2-ylmethyl]urea
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-[4-(1-benzofuran-3-carbonyl)piperazin-1-yl]benzonitrile
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyrazin-2-yl)ethan-1-one
(4S)-4-acetamido-5-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-5-oxopentanamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-methoxy-N-(pyridin-3-ylmethyl)acetamide