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N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]oxolane-3-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)furan-2-carboxamide
N-(3-methoxyphenyl)-3-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]propanamide
2-[5-(4-cyano-1-methyl-1H-pyrrol-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl]acetamide
2-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}-1,3-benzoxazole
ethyl 2-[4-(piperidine-1-carbonyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
(2S,4S,5R)-4-[(3,3-dimethylbutyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(1R,9aR)-1-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(thiophen-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(3-chlorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-methyl-2-phenylfuran-3-carboxamide
3-(2,2-diethylcyclopropanecarbonyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1S,6R)-3-methyl-9-[4-methyl-6-(methylamino)pyrimidin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(1H-imidazol-1-ylmethyl)-3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazole
2-(4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenol
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-ol
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
(2S,4R)-4-amino-1-[3-(prop-2-en-1-yloxy)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[2-(dimethylamino)ethyl]-3-(oxolan-2-ylmethyl)-1-[4-(1H-pyrazol-1-yl)phenyl]urea
N-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
1-[2-(2-fluoro-4-methylphenyl)pyridine-4-carbonyl]-4-methylpiperazine
(3S,4R)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3,5-dimethyl-4-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
2-[(2-fluorophenyl)methyl]-6-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,5-dimethyl-1,3,4-oxadiazol-2-amine
(4aS,8aR)-6-(5-ethylthiophene-3-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
{2-fluoro-5-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]phenyl}methanol
6-fluoro-2-(pyrimidin-5-yl)-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
2-(1-ethylpiperidin-4-yl)-N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]acetamide
(2S,4R)-N-ethyl-4-(2-hydroxyacetamido)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
2-(furan-2-yl)-5-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidine
1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]azocane
1-(5-{[(furan-3-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
(1S,5S)-3-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4-chloro-2-methylphenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N4-(furan-2-ylmethyl)-N1-(5-methyl-4H-1,2,4-triazol-3-yl)piperidine-1,4-dicarboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
ethyl 4-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]-1H-pyrazole-3-carboxylate
1-(furan-3-carbonyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepane
3-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-3-yl}benzoic acid
1-ethyl-N-[(2-fluorophenyl)methyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-methyl-4-(2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine-4-carbonyl)piperazine
3-(2,1,3-benzothiadiazol-4-yl)-1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]urea
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[3-(2,4-dimethylphenoxy)propyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(dimethyl-1,2-oxazol-4-yl)methyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
N-(1-cyanocyclohexyl)-2,6-dimethylpyrimidine-4-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
1-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-amine