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(1S,5R)-3-[2-(morpholin-4-yl)-2-oxoethyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(4-methyl-6-{[3-(1H-1,2,3-triazol-1-yl)propyl]amino}pyrimidin-2-yl)amino]phenol
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
2-(2-hydroxy-5-methylphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
N-(4-phenylbutyl)imidazo[1,2-a]pyridine-6-carboxamide
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1-methyl-1H-indazol-3-yl)-2-[3-(pyridin-3-yl)-1H-indazol-1-yl]acetamide
8-methoxy-4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[(2-chloropyridin-3-yl)methyl]-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
4-[6-(piperazin-1-yl)pyridin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-benzyl-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecane
4-(2-aminopyridine-4-carbonyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
2-[2-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-pyrrol-1-yl]-1,3-thiazole
N-cyclopropyl-3-[5-(pyridine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
2-[1-benzyl-5-(4-methyl-3-oxo-3,4-dihydroquinoxalin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
8-(butan-2-yl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-8-[(3-hydroxyphenyl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methyl-3-(pyrrolidin-1-ylmethyl)-1,2-dihydroquinolin-2-one
4-(4-methylphenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
N-[4-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)carbamoyl)phenyl]-2-methylfuran-3-carboxamide
1-{9-[2-(benzyloxy)ethyl]-3,9-diazaspiro[5.5]undecan-3-yl}-3-methoxypropan-1-one
2-{[(1,4-dimethylpiperidin-4-yl)methyl][(2E)-3-phenylprop-2-en-1-yl]amino}ethan-1-ol
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(carbamoylmethyl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-3-carboxamide
N-[(2S)-2-aminopropyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(3,5-dimethylphenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
2-amino-4-(5-tert-butyl-1H-pyrazol-3-yl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
3-ethyl-8-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentyl-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
5-{methyl[2-(methylcarbamoyl)ethyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3S,4S)-1-(7-chloro-4-hydroxyquinoline-3-carbonyl)piperidine-3,4-diol
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2-(pyrrolidin-1-yl)benzamide
(2S,4S)-4-(4-{[1-(3-chloro-2-fluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-1-yl)ethan-1-ol
(4aR,8aR)-4-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-octahydro-2H-1,4-benzoxazine
(1R,5R)-6-(2-methoxypyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
5-(1-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
6-fluoro-4-(4-methanesulfonylphenyl)-1,3-benzothiazol-2-amine
3-({2-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
6-methoxy-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
2-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-3-carboxamide
2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxo-N-phenylacetamide
1-methyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine