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1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(4-{[3-(methylsulfanyl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1-(4-methoxyphenyl)-6,6-dimethyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)-5-phenyl-1,2-oxazole-3-carboxamide
3-cyclopropyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-(1H-imidazol-2-yl)-1-[3-(5-methylfuran-2-yl)benzoyl]piperidine
N-{4-oxo-4-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butyl}acetamide
3-benzyl-5-{[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl}-1,2,4-oxadiazole
(3R,4S)-4-({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)amino)oxolan-3-ol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
4,4-difluoro-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
1-methyl-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2-phenylpiperazine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-4-(hydroxymethyl)-N-methylpyridine-2-carboxamide
2-[3-(methoxymethyl)phenyl]-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-methylprop-2-en-1-yl)piperidine
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
N-ethyl-6-(2-fluorophenyl)-N-(oxolan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(2-methoxyethyl)-2-methyl-3-({[(1R)-1-phenylpropyl]carbamoyl}amino)benzamide
3-{1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(3,3-difluoropiperidin-1-yl)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
8-methoxy-2-methyl-4-(5-phenoxyfuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N,N-dimethylpyridine-3-carboxamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}cycloheptanamine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1-[(4-methoxyphenyl)methyl]-1H-pyrazole
3,5-dimethyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2-oxazole-4-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-{1-[5-(2-chlorophenyl)furan-2-carbonyl]azetidin-3-yl}pyridine
(3R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]pyrrolidin-3-ol
1-(3-methoxyphenyl)-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
8-[(3,5-dimethylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-(2-hydroxyethyl)-2-(3-phenyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3,5-dimethyl-1H-indole-2-carboxamide
5-[3-(1H-imidazol-2-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N,4-dimethyl-6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidin-2-amine
2-amino-7-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-[2-(benzyloxy)ethyl]-N,N-dimethyl-2,7-diazaspiro[4.5]decane-2-carboxamide
(1S,5R)-6-[(5-methylthiophen-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,5-dimethoxyphenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
2-(4-fluorophenyl)-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]morpholine
1-butyl-4-{1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazin-2-one
N-(2,3-dimethylphenyl)-N'-[2-hydroxy-3-(3-methoxyphenoxy)propyl]propanediamide
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
(2S,4R)-4-(dimethylamino)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxylic acid
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-methylpyrimidin-4-ol
[1-(5-chloropyridin-2-yl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
(3aR,6aS)-5-(2-cyanobenzoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid