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7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-methanesulfonylacetamide
(1R,5R)-N-(3,4-difluorophenyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-methoxybenzoic acid
ethyl 1-(1H-pyrazol-3-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(2-phenoxyethyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}acetamide
6-ethyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
(3aS,6aS)-2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-oxo-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-2-(morpholin-4-yl)benzamide
3-[4-(6-methoxypyrimidin-4-yl)piperazin-1-yl]pyrazine-2-carbonitrile
4-(5-methylpyridin-2-yl)-1-[(2,4,6-trimethylphenyl)methyl]piperidin-4-ol
2-ethyl-4-methyl-5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-imidazole
2-cyclopropyl-6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-benzoxazole
2-{[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]methyl}pyridine-3-carboxylic acid
ethyl 4-(2-phenoxyethyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
4-(2,4-dimethylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}cyclopropane-1-carboxamide
N-(2-methoxyethyl)-N,5-dimethyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-butyl-5-methyl-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-ethoxyethyl)-3-[methyl(1-methylpyrrolidin-3-yl)sulfamoyl]benzamide
6-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}pyridine-2-carboxylic acid
2-{4-[2,2-dimethyl-3-(morpholin-4-yl)propyl]morpholin-2-yl}ethan-1-amine
4-({1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)piperazin-2-one
methyl 1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
3-(dimethyl-1,2-oxazol-4-yl)-N-(1,2-oxazol-3-ylmethyl)propanamide
4-({3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2,3,6-tetrahydropyridine
(4aR,8aR)-2-methanesulfonyl-7-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
3-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]urea
1-methyl-4-(4-methylpyrimidin-2-yl)-1,4,9-triazaspiro[5.5]undecane
5-({[2-(trifluoromethoxy)phenyl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
(benzylsulfamoyl)({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
2-[4-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)phenyl]acetic acid
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-amino-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5,6-dimethyl-2-oxo-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
5-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[2-(2-methylpropanesulfonyl)ethyl]quinoxaline-5-carboxamide
(2S)-N-(3-chloro-2,6-dimethylphenyl)-2-(piperidine-1-carbonyl)pyrrolidine-1-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(1H-indazol-1-yl)propyl]propanamide
methyl 2-{1-[(3-chloro-4-fluorophenyl)carbamoyl]pyrrolidin-3-yl}acetate
N-methyl-N-(3-phenoxypropyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidin-2-amine
4-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
6-{[3-(4-hydroxypiperidin-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(1H-imidazol-2-ylmethyl)-3-(2-phenylethyl)piperidine
1-(1-methyl-5-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol