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3-(dimethylamino)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)benzamide
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
5-acetyl-N-methyl-N-(2-methylprop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
{1-[(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-N-methyl-3-phenylpropanamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2,5-difluorophenyl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-{1-[2-(morpholin-3-yl)acetyl]piperidin-4-yl}propanamide
ethyl 4-[(4-{[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
2-[3-(trifluoromethoxy)phenyl]benzamide
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-ethyl-N-(2-methylphenyl)propanamide
1-[2-(1H-pyrazol-1-yl)acetyl]-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
2-phenyl-4-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
5-{[2-(dimethylamino)ethyl](methyl)amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
6-[6-hydroxy-4-(3-methoxypropanoyl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-(3-propylmorpholin-4-yl)ethan-1-one
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-(1H-imidazol-2-yl)piperidine
6-methoxy-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
2-amino-6-hydroxy-4-(thiophen-3-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
1-(cyclopropylmethyl)-N-methyl-5-(1-methylpiperidine-2-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-ethoxypropan-1-one
1-(5-ethylthiophene-3-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
4-(1H-1,3-benzodiazol-1-yl)-1-(furan-3-carbonyl)piperidine-4-carboxylic acid
N-(1-{[4-hydroxy-3-(prop-2-en-1-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
2-methyl-5-propyl-4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)pyrimidine
5-methoxy-2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4H-pyran-4-one
methyl[(2E)-2-methylbut-2-en-1-yl]{[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-(1-cyclopropanecarbonylpiperidin-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
3-(2-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl)pyridine
N-{[1-(3,4-difluorobenzoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
ethyl 1-(cyclopropylmethyl)-5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-{[3-(1H-indol-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
2-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
(4S)-1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-4-carboxamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
2-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]benzamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopropane-1-carboxamide
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
(cyclohexylmethyl)[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-(2-methoxy-5-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetic acid
4-(4-chlorophenoxy)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-hydroxyethan-1-one
N-[(5-chloro-2-fluorophenyl)methyl]-N,2,2-trimethyloxan-4-amine