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1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-hydroxypiperidine-4-carboxylic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
5-methyl-1-(2-methylphenyl)-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperazin-2-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
5-oxo-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}propanamide
3-{2-oxo-2-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}imidazolidine-2,4-dione
2-(ethylsulfanyl)-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-phenyl-N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]benzamide
4-(1H-indol-3-yl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]butan-1-one
N-benzyl-5-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}pyrimidin-2-amine
3-acetamido-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)propanamide
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-1-[1-(piperidine-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
5-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
8-(furan-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{[6-(dimethylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}-2-methylheptan-2-ol
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-(morpholin-4-yl)butan-1-one
4-(4-oxo-4H-chromen-3-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(3R,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[3-(1-methoxyethyl)phenyl]-N,N-dimethylbenzamide
8-fluoro-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]quinoline-2-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-N-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-(1,2-oxazinan-2-yl)pyridine-3-carboxamide
1-{5-methyl-2-[(propan-2-yl)amino]benzoyl}piperidine-4-carboxamide
N-(4-{4-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]piperidin-1-yl}phenyl)-2-phenoxyacetamide
(4aR,7aS)-4-[(3-fluoro-4-methoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]benzonitrile
5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-methoxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
3-(1-methoxypropan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-ethyl-5-(1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-methoxyethyl 2-methyl-2,8-diazaspiro[4.5]decane-8-carboxylate
2-(3-hydroxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
3-methyl-5-(1H-pyrazol-3-yl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
3-cyclopropyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1H-pyrazole-5-carboxamide
2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-9-oxa-2-azaspiro[5.5]undecane
N-methyl-2-(pyridin-4-ylsulfanyl)-N-(quinolin-6-ylmethyl)acetamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propane-1,2-dione
3-[2-(3,4-dichlorophenyl)morpholin-4-yl]propanamide
7-acetamido-N-methyl-N-[2-(oxan-2-yl)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-ol
3-(cyclopropylmethyl)-N-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide