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2-[({1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
5-(2-amino-2-methylpropanoyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(2-methylphenyl)methyl]amino}butan-1-ol
2-(4-chloro-2-methylphenoxy)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
4-[(2,4-dimethylphenyl)methyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
4-(2,5-dimethoxyphenyl)-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4H-1,2,4-triazole
1-(4-{4-[(3-hydroxypyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
5-methanesulfonyl-N-[(3-methoxyphenyl)methyl]-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
5-(morpholin-4-ylmethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}furan-3-carboxamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
(2S)-3-[1-(5-chloropyridin-2-yl)-1H-imidazol-4-yl]-2-acetamidopropanoic acid
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(propan-2-yl)piperidin-4-ol
2-(1-{2-[4-(methylsulfanyl)phenyl]ethyl}piperidin-4-yl)propan-2-ol
2-(dimethylamino)-N-{3-methyl-1-[7-(5-methylthiophene-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
4-methyl-5-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
6-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[2-hydroxy-1-(thian-4-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methanol
(4aR,8aR)-2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-7-cyclopentanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
5-(furan-2-yl)-3-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylacetamide
1-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
(3R,4S)-1-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-4-phenylpyrrolidin-3-amine
(3S,4R)-1-[(6-chloropyridin-3-yl)methyl]-3-ethyl-4-methylpiperidin-4-ol
3-(1-butyl-1H-imidazol-2-yl)-1-(pyrrolidine-1-sulfonyl)piperidine
2-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)acetamide
N4-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-6-methylpyrimidine-2,4-diamine
2-chloro-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
(3S,4S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
8-methoxy-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]oxy}pyridine
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,1-benzoxazole-3-carboxamide
1-(but-3-enoyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)-2,2-dimethyloxane-4-carboxamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{[1-(pyridine-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
propan-2-yl 4-chloro-3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}carbamoyl)amino]benzoate
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2,4,5-trimethoxyphenyl)methyl]amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1H-1,2,4-triazol-3-ylmethyl)acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-cyclopentyl-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpropanamide
N-[(2S,4R,6S)-2-benzyl-6-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]oxan-4-yl]acetamide
4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane