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5-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-methyl-N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
dimethyl(3-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}propyl)amine
(2R)-2-({[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}amino)-2-phenylethan-1-ol
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-2-one
2-{3-[2-(3-methoxyphenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
6-{2-[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
2-(3-chlorophenyl)-N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
2-amino-4-(4,5-dimethylfuran-2-yl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
1-[(1S,5R)-6-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]methyl}-3-phenylpropanamide
3-[({[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}carbamoyl)amino]-N,N,2-trimethylbenzamide
5-(methoxymethyl)-N-[3-methyl-1-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]furan-2-carboxamide
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2,2-difluoro-N-({1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}methyl)acetamide
1-[1-(2H-1,3-benzodioxol-5-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
2-(2-methoxyethyl)-8-(6-methylquinolin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-hexyl-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(pyrazin-2-yl)propan-2-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-benzyl-5-[1-(propan-2-yl)-1H-imidazol-2-yl]pyrimidin-2-amine
5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-N-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidine
3-{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
N-(1-benzothiophen-5-ylmethyl)-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
(3S,4S)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
2-(1H-1,3-benzodiazol-1-yl)-N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]acetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-amino-N-({1-[(3-ethenylphenyl)methyl]piperidin-3-yl}methyl)cyclobutane-1-carboxamide
1-(dimethylamino)-3-(4-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
1-(4-{[2-(morpholin-4-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N,N-dimethyl-2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-(3-chloro-4-methoxyphenyl)-N-cyclopropylpyridine-4-carboxamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-9-oxa-2-azaspiro[5.5]undecane
N-cyclopentyl-1-(3-methylbutyl)-4-oxo-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
4-(3-methyl-1,2-benzoxazol-5-yl)-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1-[3-(1,3-oxazol-5-yl)phenyl]urea
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
1-({4-[4-(1-methoxyethyl)phenyl]phenyl}methyl)piperazine
8-[3-(1H-imidazol-1-yl)butanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N'-(3-chloro-4-fluorophenyl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)propanediamide
4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]thiomorpholine
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(methylamino)acetamide
3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
6-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]pyrazine-2-carboxamide
3-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}aniline