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N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
ethyl 3-{[5-(cyclooctylcarbamoyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridin-3-yl]formamido}propanoate
3-(4-chloro-2-methylbenzoyl)-1-(oxan-4-yl)piperidine
(2E)-N-{[3-methyl-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
2-methyl-5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,4-dihydropyridin-4-one
N-(quinolin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-5-[(methylsulfanyl)methyl]-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
3-[(2-oxopiperidin-3-yl)sulfamoyl]-N-phenylbenzamide
1-{2-[5-(1-ethyl-3-methylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
2-(5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}furan-2-yl)benzonitrile
4-(5-methoxypyrimidin-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-benzyl-N-methyl-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-cyclopropyl-6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
1-[2-(3,4-dimethoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(2-methylpropyl)piperidine-3-carboxamide
(4aR,8aR)-2-methanesulfonyl-7-(6-methylpyridazin-3-yl)-decahydro-2,7-naphthyridin-4a-ol
5-(1-benzothiophene-5-carbonyl)-3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
N-{3-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-oxopropyl}methanesulfonamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}[(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
2-(3-methoxypropyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-cyclopropyl-N-(2-ethoxyphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(2-methoxyethyl)-4-({[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}methyl)pyrrolidin-2-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-propylpiperazine
2-methoxy-1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
5-propyl-1'-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperazin-1-yl)isoquinoline
4-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-2-amine
3-[3-(2,5-difluorobenzoyl)piperidine-1-carbonyl]-2-methoxypyridine
1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-[2-(propan-2-ylsulfanyl)phenyl]urea
(1S,4S)-5-[(4-ethylphenyl)methyl]-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-3-phenoxypropanamide
dimethyl[(4-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}-1,3-thiazol-2-yl)methyl]amine
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]pyrimidine-5-carboxylic acid
4-(4-chloro-1H-pyrazole-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-(6-chloro-2H-chromene-3-carbonyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
2,6-dimethyl-3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
1-(4-{7-chloro-3-[(cyclooctylamino)methyl]quinolin-2-yl}piperazin-1-yl)ethan-1-one
2-(1H-pyrazol-1-ylmethyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1,4-oxazepane-4-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
5-cyclobutyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,3,4-oxadiazol-2-amine
5-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-1H-1,2,3-benzotriazole
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine