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N-[(3S,4R)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(3R,4R)-4-ethyl-1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)piperidine-3,4-diol
1-(3,4-dimethylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-6-methyl-3,4-dihydroquinazolin-4-one
1-(2-methoxyethyl)-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethyl-1,3-oxazole-4-carboxamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(oxolane-2-carbonyl)piperazine
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(4-fluorophenyl)morpholine
1-(4-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidin-1-yl)ethan-1-one
3-[(3R,4S)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(2-methylphenyl)piperazine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]propanamide
(3R,5S)-N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
(1S,5R)-6-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-methanesulfonyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N3-[2-(3-chlorophenyl)ethyl]-N5-cyclopentyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(cyclopentyloxy)phenyl]-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
N-(2-methoxyethyl)-1-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
N-ethyl-2-[(2-fluorophenyl)methyl]-1,6-dimethyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(3aR,6aS)-1-oxo-5-{[3-(trifluoromethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
(1S,5R)-3-(1,3-benzoxazol-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-chloro-5-acetamido-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]benzamide
N-methyl-2-(4-{4-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]butanoyl}morpholin-3-yl)acetamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1R,5S)-3-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-4-(3-fluorophenyl)-1-(4-hydroxybenzoyl)pyrrolidine-3-carboxylic acid
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
N-benzyl-1-methyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{3-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-5-cyclopropyl-1,3-oxazole
N-(2-methoxyethyl)-1-methyl-N-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-amine
2,2-dimethyl-N-({1-[(8-methylquinolin-5-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-hydroxybutan-2-yl)-1,3-oxazole-4-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(1-methylpiperidin-4-yl)-2-phenylacetamide
1-ethyl-6-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-indole
3-benzyl-1-methyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenoxy)acetamide
4,5-dimethyl-6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
1-ethyl-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-(2-hydroxyethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(1,3-thiazole-4-carbonyl)piperidine
methyl 6-[(2-fluoro-4-methoxyphenyl)methyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-benzyl-4-(7-fluoro-2-methylquinoline-4-carbonyl)piperazin-2-one
4-methyl-N-(3-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)benzamide
7-(2-propyl-1,3-thiazole-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide