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1'-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-hydroxy-2-(pyridin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidine-5-carboxamide
3-[2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-(2H-1,3-benzodioxol-5-yl)-5-(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazole
1-methyl-3-[4-(4-{[(3-methyl-1H-pyrazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
2-(2-{[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
N-(1,3-dihydroxypropan-2-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
(1S,4S)-2-(2-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}ethyl)-2-azabicyclo[2.2.1]heptane
[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-chloro-1,2-dihydropyridin-2-one
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-fluoroquinolin-3-yl}methyl)[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
N-(2-hydroxyethyl)-1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3,5-dichloro-4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}pyridine
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-cyclopentyl-1-methyl-5-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
5-ethyl-2-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]pyridine
9-(2,4-difluorobenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1,3-oxazole
2-({5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
1-[(2,6-difluorophenyl)methyl]-N-(furan-3-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)-1λ6-thiolane-1,1-dione
1-(4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-1H-pyrazole
5-fluoro-2-[3-(pyridin-2-yl)azetidin-1-yl]pyridine
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,5-dimethylpyrazine
2-cyclopentyl-N-(3-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(pyridin-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl[(4-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}phenyl)methyl]amine
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-ethyl-4,5-dihydro-1,2-oxazole
6-(3,4-dimethylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-{5-[(2S)-1-methanesulfonylpyrrolidine-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
2-propyl-5-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
7-{[4-(2-hydroxyethoxy)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(adamantan-2-yl)-1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-methoxy-N-({5-[(4-methoxy-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-ethyl-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
6-ethoxy-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
8-[(2-ethoxyphenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(benzylsulfamoyl)(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)amine
3-(2-hydroxyphenyl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}propan-1-one
1-[(3-methoxyphenyl)methyl]-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperazin-2-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-{5-[2-(2-oxopyrrolidin-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid