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N-ethyl-4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxamide
4-[3-(furan-2-yl)phenyl]-4H-1,2,4-triazole
4-{4-[(1-benzothiophen-2-ylmethyl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2,4-dichloro-3-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}phenol
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(4-methoxyphenyl)piperazine
dimethyl[(5-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}thiophen-3-yl)methyl]amine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(butan-2-yl)-6-methyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(cyclopropylmethyl)-2-(4-fluorophenyl)-N-(2-methoxyethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-[1'-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-N-(1,2-oxazol-3-ylmethyl)propanamide
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-[(4-chlorophenyl)methyl]-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-4-[7-(5-methyl-1,3-oxazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazine
N-(4-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenyl)acetamide
N-(1-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-3-carboxamide
1-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[4-(1H-pyrazol-1-yl)butan-2-yl]urea
2-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetic acid
(1R,3S)-3-(2-aminoethoxy)-7-[4-(5-methylfuran-2-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
(3R,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-methoxy-5-[1-(quinoxalin-6-yl)-1H-imidazol-2-yl]phenol
(1R,7S)-N-methyl-3-(3-methylbutyl)-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
8-(4-methyl-1H-pyrrole-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxybenzoyl)piperidine
(2S,4R)-4-amino-N,N-diethyl-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
4-[2-(2-methoxyethoxy)acetyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-6-methylquinolin-4-ol
3-[(3R,4S)-4-(dimethylamino)-1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]propan-1-ol
ethyl 4-{4-[2-(phenylcarbamoyl)ethyl]piperidin-1-yl}piperidine-1-carboxylate
N-{[2-(diethylamino)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
N-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}methanesulfonamide
5-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pentan-1-ol
1-(3-chloro-4-ethoxyphenyl)-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
6-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]pyrimidin-4-amine
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-[4-(4-chlorophenyl)-1H-imidazol-2-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
1-{3-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-ethyl-N-[1-(4-methylpyridin-2-yl)propyl]pyrimidine-5-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
6-methyl-3-(2,3,4-trimethoxyphenyl)pyridin-2-amine
N-(1-ethyl-1H-indazol-3-yl)-2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetamide
N-[2-(1H-indol-3-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(2S,4S)-4-amino-1-[3-(2-methoxyphenyl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(3S,5S)-1-(2-cyclohexylethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
2-{[4-(2-methylphenyl)-5-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-(2-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-ethyl-4-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}pyrimidine