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4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
2,5-dioxo-6-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
methyl 1-{[4-(phenylamino)quinazolin-2-yl]methyl}piperidine-2-carboxylate
N-[1-(furan-2-carbonyl)piperidin-3-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propanamide
(4-{[(2-amino-9H-purin-6-yl)(methyl)amino]methyl}oxan-4-yl)methanol
1-(3-chloro-4-methoxyphenyl)-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
methyl(3-phenylpropyl)(pyrazin-2-ylmethyl)amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(pyridin-2-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
3-hydroxy-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
ethyl 1-(4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzoyl)piperidine-4-carboxylate
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-phenoxyethan-1-one
5-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1,3,4-oxadiazol-2-amine
6-{1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]piperidin-3-yl}-2-methyl-3,4-dihydropyrimidin-4-one
N-(1,3-benzoxazol-2-ylmethyl)-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(1R,5R)-N,N-dimethyl-6-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-(dimethylamino)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-[(2R)-3-methylbutan-2-yl]piperidine-1-carboxamide
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-hydroxyethyl)-N-methylacetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}propanamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-methylpyrimidin-2-amine
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
6-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)sulfanyl]propan-1-one
2-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
3-(3-methoxypropyl)-1-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxylic acid
1,3-dimethyl-5-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
ethyl 1-[(2-aminopyrimidin-5-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N,N-dimethyl-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
3-methyl-7-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
6-fluoro-8-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]quinoline
(1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)methanol
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-ethyl-3,5-difluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-2-carboxamide
2,3-dimethoxy-N-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]benzamide
6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
[(2,3-dimethoxyphenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(propan-2-yl)amine
2-{[5-(2,2-dimethylcyclopropyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl](3-chlorophenyl)methanol
1-[2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
(1R,5R)-3-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane