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(3R,4R)-N-cyclohexyl-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[4-oxo-4-(3-phenylpiperazin-1-yl)butyl]pyrrolidin-2-one
2-(2-aminoethyl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
1-ethyl-4-[(2-phenylphenyl)methyl]piperazine-2,3-dione
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[4-(3-acetylphenyl)phenyl]-3-[(1R,2S)-2-hydroxycyclohexyl]-3-methylurea
N-[2-(4-chlorophenyl)ethyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)acetamide
4-(2-methoxyphenoxy)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxylic acid
1-(4-{[4-(hydroxymethyl)-4-methylpiperidin-1-yl]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethoxy]ethan-1-ol
methyl (1R,3S,3aR,6aS)-5-ethyl-3-(1-methyl-1H-imidazol-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-{1-[3-ethoxy-4-(prop-2-en-1-yloxy)phenyl]-N-(propan-2-yl)formamido}propanamide
methyl 5-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-[4-(pyridin-2-yl)pyrimidin-2-yl]thiomorpholine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]sulfonyl}-1H-pyrazole
1-methyl-6-propyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}propan-1-one
(2R)-2-hydroxy-N-methyl-2-phenyl-N-(quinoxalin-2-ylmethyl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(pyrazine-2-carbonyl)-1,4-diazepane
1-methyl-3-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-1-[3-(oxolan-2-yl)propyl]urea
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-(methoxymethyl)-6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanamide
2-methyl-N-{1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-[(2-chlorophenyl)methyl]-4-[4-(furan-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclooctyl-2-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}acetamide
N-ethyl-5-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
1-[4-(difluoromethoxy)benzoyl]-3-(2-methylphenoxy)azetidine
1-(4-acetylphenyl)-3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]urea
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methylfuran-3-carboxamide
{[5-(oxan-2-yl)furan-2-yl]methyl}(propyl)(pyridin-3-ylmethyl)amine
4-[4-(azetidine-1-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
1-[1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-(adamantan-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]acetamide
(4-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}oxan-4-yl)methanol
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
1'-{[3-(cyclopentyloxy)phenyl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carboxylic acid
6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carboxamide
1-(3-chloro-4-methoxybenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(1S,5R)-6-benzyl-3-(1-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one