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4-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
(3R,4R)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(pyridin-2-ylformamido)methyl]benzoate
N-[(3R,4S)-4-cyclopropyl-1-[(methylcarbamoyl)methyl]pyrrolidin-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
(1R,5S,6R,7S)-N,3-dimethyl-4-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-cyclopropyl-1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[2-(pyridin-2-yl)ethyl]amino}pyrimidine-5-carboxylic acid
(1S,4S)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2-(2-methyl-1,3-benzothiazol-5-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(2H-1,3-benzodioxol-5-yl)-2-(pyrrolidin-1-yl)acetic acid
4-(2,1,3-benzoxadiazol-4-yl)-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-methoxy-N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
2-methyl-N-{4-methyl-2-[3-(pyrazin-2-yl)propanamido]phenyl}benzamide
1-[4-(difluoromethoxy)phenyl]-3-[3-(4-methylpiperazin-1-yl)propyl]urea
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
2-(3-methoxypropyl)-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine
3-({2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
4-[(4-fluorophenyl)methyl]-1-(furan-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-[1-(3-fluoro-4-methylbenzoyl)-4-phenylpiperidin-4-yl]ethan-1-one
4-[3-(3-benzylpyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyrimidin-2-amine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-3-ylmethyl)amine
1'-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]spiro[indene-1,4'-piperidine]
3-(1,2-oxazinan-2-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
(1R,5S,6R,7S)-6-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-3-methyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-methyl-3-(1-propyl-1H-1,3-benzodiazol-5-yl)-1-[1-(pyridin-3-yl)pentyl]urea
3-{[3-(benzyloxy)piperidin-1-yl]methyl}-6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2,5,7-trimethylquinoline
5-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidin-3-ol
3-(2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-2-yl}ethyl)phenol
1-[(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}thiophen-3-yl)sulfonyl]pyrrolidine
4-chloro-5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
2-[4-(dimethylamino)phenyl]-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
ethyl 4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamido]piperidine-1-carboxylate
[(3R,4R)-1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
N-[(4-chlorophenyl)methyl]-2-(2-hydroxypropanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(1-ethyl-1H-indazol-3-yl)-2-{4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
7-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
5-(4-methyl-1,4-diazepan-1-yl)-2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
1-(2-methoxy-5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane