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1-{5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-1,4-diazepan-5-one
N-methyl-1-[(3-phenoxyphenyl)methyl]piperidine-2-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
4-[3-methyl-5-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
N-{3-[({3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}carbamoyl)methoxy]phenyl}propanamide
5-(2-chloro-4-fluorophenoxymethyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide
1-({1-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
ethyl 4-{[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]amino}piperidine-1-carboxylate
methyl 3-[(3S,4R)-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-1-[(3-phenoxyphenyl)methyl]piperidin-3-yl]propanoate
[1-(2-cyclopropylpyrimidine-5-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
2-(2-{[2-(2-methylpropanamido)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
methyl[(6-methylpyridin-2-yl)methyl][2-(oxan-4-yl)ethyl]amine
(3R,4R)-4-(azepan-1-yl)-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-3-ol
8-[2-(2-chloro-6-fluorophenyl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)acetate
(4aS,8aR)-6-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(2,4-difluorobenzoyl)-3-(3-methoxyphenoxymethyl)piperidine
4-(4-fluorophenoxy)-1-(furan-3-carbonyl)piperidine-4-carboxylic acid
4-(5-methylpyridin-2-yl)-1-[6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-ol
4-[4-(2-chloro-4-fluorophenyl)phenyl]piperidin-4-ol
5-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridine-2-thiol
1-(3-phenylbutyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(carbamoylmethyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidine-3-carboxamide
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-6-ethoxyphenol
1,9-dimethyl-4-(quinoxaline-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(benzenesulfonyl)-7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(dimethylamino)-N-[2-(ethanesulfonyl)ethyl]-2-(3-methylphenyl)acetamide
(2S,4R)-4-amino-N-ethyl-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-[2-(1H-indazol-3-yl)acetamido]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)-1λ6-thiolane-1,1-dione
2-{1-[(4-ethoxyphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(1R,3S,5S)-3-(4-methoxyphenyl)-8-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-8-azabicyclo[3.2.1]octane
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(1,3-thiazole-4-carbonyl)-1,4-diazepan-5-one
6-[(3aS,6aS)-1-(piperidine-1-carbonyl)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1,3-benzothiazole
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
2-[(2S)-2-aminopropanoyl]-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3S,4R)-1-(4-chloro-2-fluorobenzoyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-amino-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-3-carboxylic acid
methyl[(5-methylfuran-2-yl)methyl]({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
2-benzyl-8-(furan-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,3-dihydro-1-benzofuran-5-carboxamide
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-8-methyl-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-5-methyl-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-1H-pyrazole-4-carboxamide