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N-[1-(1H-imidazol-2-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-4-carbonitrile
2-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-2,3-dihydro-1H-isoindole
ethyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
7-fluoro-3-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}-1,2-dihydroquinolin-2-one
(1-benzothiophen-2-ylmethyl)(methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(oxolan-3-ylmethyl)-3-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]-2-ethylpyridine-4-carboxamide
N-{4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-oxobutyl}acetamide
4-[2-({4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-5-methylpyrimidin-2-yl}sulfanyl)ethyl]morpholine
4-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-4-yl}pyridine
1-[cyclopropyl(4-methoxyphenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
2-{5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[(5-methylpyrazin-2-yl)methyl]amine
2-{[(3S)-3-hydroxypyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[5-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
5-oxo-N-(2-phenylphenyl)-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-methylpropan-1-one
1-[3-(1H-imidazol-1-yl)propyl]-5-(2-methylpropyl)-4-phenyl-1H-imidazole
4-methyl-2-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-amino-6-(5-chlorothiophen-2-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
4-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyrimidin-2-amine
1-{[1-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
3-(3-fluorophenyl)-4-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]acetamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
1-ethyl-4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[1-({1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)piperidin-4-yl]acetamide
3-[2-(methylsulfanyl)benzoyl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
ethyl 4-oxo-5-phenoxy-1-[4-(pyrrolidin-1-yl)butyl]-1,4-dihydropyridine-3-carboxylate
1-[2-(4-methoxyphenyl)ethyl]-5-(oxane-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-1-({[4-(pyridin-2-ylmethoxy)phenyl]carbamoyl}amino)cyclohexane-1-carboxamide
(4aS,7aR)-4-(1H-1,3-benzodiazol-2-ylmethyl)-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methanol
(4-phenyl-5-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(3,5-dimethylphenyl)-4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-2-one
1-(2-methoxyethyl)-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
(4aS,7aR)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-ethoxy-2-fluorophenyl)-3-[3-(1H-imidazol-2-yl)propyl]urea
1-({1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-[3-(benzyloxy)propyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-pyrrole-3-carboxamide
3,3-dimethyl-1-[(3S,4R)-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea