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1-ethyl-3-methyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
N-{1-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
1-(2-methylpyridin-4-yl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane
4-benzyl-3-ethyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
N-ethyl-1-(5-fluoro-1H-indole-2-carbonyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-(oxan-4-yl)piperidine-3-carboxamide
3-[2-(dimethylamino)-4-methylpyrimidine-5-amido]pyrrolidine-3-carboxylic acid
methyl[(5-methylfuran-2-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-{1-oxa-8-azaspiro[4.6]undecan-8-yl}propan-1-one
N-(4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopentanecarboxamide
8-(2,8-dimethylquinoline-3-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-methyl-2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane
N-[(3,5-difluorophenyl)methyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1-methyl-1H-pyrazole-4-carboxamide
1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}-N,N-dimethylpyrrolidin-3-amine
3-chloro-6-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)pyridazine
{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
1-{5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
5-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}quinoline
1-[(3,5-dimethoxyphenyl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
2-(3-fluorophenyl)-2-[(5-propyl-1,2-oxazol-3-yl)formamido]acetic acid
N-[1-(2-methylphenoxy)propan-2-yl]-N'-(4-methylphenyl)propanediamide
4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,4-oxazepan-6-ol
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}benzamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
4-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-1,4-oxazepan-6-ol
1-[2-(1H-pyrazol-3-yl)phenyl]piperazine
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
ethyl 4-{2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazine-1-carboxylate
N-[2-(2,3-dichlorophenyl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-(2-oxoazepan-1-yl)acetamide
5,6-dimethoxy-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,2-dihydroisoquinolin-1-one
4-(2-fluoro-5-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidine
3-[1-(2,6-dimethoxypyrimidin-4-yl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
N-[2-(2,4-difluorophenyl)-1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}-6-(pyrrolidine-1-carbonyl)pyrazine
4-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl}benzoic acid
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
6-methyl-5-(2-phenylphenyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
(3S,4S)-1-[4-(hydroxymethyl)benzoyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
(isoquinolin-5-ylmethyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(adamantan-1-yl)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazine
N-(2-methoxyethyl)-5-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide