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2-methoxy-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)benzoic acid
7-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-2-ethyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
3-ethyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,4-oxadiazole
1-ethyl-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
3-methyl-N-[1-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(oxan-4-yl)-decahydro-1,6-naphthyridin-2-one
3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
2-{4-[2-(adamantan-1-yl)acetyl]morpholin-3-yl}acetic acid
5-methanesulfonyl-2-methyl-N-[1-(6-methylpyridin-2-yl)propyl]pyrimidin-4-amine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxy-N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
(4aS,7aR)-1-(2-ethylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1H-imidazol-1-ylmethyl)-1-[3-(methylsulfanyl)propyl]piperidine
3-{[6-(aminomethyl)pyrimidin-4-yl]amino}-N-(naphthalen-1-yl)propanamide
5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-N-propylpyrimidin-2-amine
9-(6-aminopyridine-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{[(3-methoxyphenyl)methyl](propyl)amino}piperidin-1-yl)ethan-1-one
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
1-[(3S,4R)-3-cyclopropyl-4-[(5-propylpyrimidin-4-yl)amino]pyrrolidin-1-yl]-2-(methylamino)ethan-1-one
2-(2,3-difluorophenoxymethyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 2-{2-[2-(cyclopentylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanoate
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-ethyl-1-benzofuran-3-yl)-1H-imidazole
(3S,4S)-4-(naphthalen-2-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
3-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
(1S,4S)-5-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(3S,5R)-N3-[3-(dimethylamino)propyl]-N5-(4-fluorophenyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N2-cyclopropyl-N5-[(3-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
6-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
3-cyclohexyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(thiophen-3-yl)propanamide
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-methylurea
methyl 6-{[methyl(oxolan-3-yl)amino]methyl}-3-(2-phenoxyacetamido)thieno[2,3-b]pyridine-2-carboxylate
5-(2,6-difluorophenyl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
1-[1-(9H-fluoren-2-ylmethyl)piperidin-3-yl]-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-({2-[butyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)-N-methylpyrrolidine-3-carboxamide
N-[4-(azepan-1-yl)butyl]-2-(3-fluorophenyl)-2-hydroxyacetamide
5-cyclopropanecarbonyl-1'-(pyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-methoxyphenyl)methyl]-1-[3-(4-methylphenyl)propanoyl]-1,4-diazepan-5-one
2-amino-6-(2-fluoro-5-methoxyphenyl)pyrimidin-4-ol
N3-cyclohexyl-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-chloro-4-({[3-oxo-3-(pyrrolidin-1-yl)propyl]carbamoyl}amino)-N-propylbenzamide