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2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(methylsulfanyl)propyl]piperidine
2-(1H-indole-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
(4S,4aS,8aR)-1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
N-[2-(furan-2-yl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[(3R,5R)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperidine
1-methyl-6-(propan-2-yl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[8-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-N,N-dimethylazepan-4-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
dimethyl[(4-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-2-yl}phenyl)methyl]amine
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
N-cyclopropyl-2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
7-methyl-2-(2,3,4-trimethoxyphenyl)-1H-1,3-benzodiazole
2-(dimethylamino)-2-(2-methylphenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
(3aS,6aS)-2-(3-cyano-2-methoxypyridin-4-yl)-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine
1-({4-[(1-methyl-1H-1,2,3-triazol-4-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[4-(1H-imidazol-1-yl)benzoyl]-4-(4-methylphenoxy)piperidine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-chloro-4-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]phenol
3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N,N-dimethyl-2-[(1S,5R)-6-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
5-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
3-(2-hydroxyethyl)-4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-2-one
3-(2-oxopiperidin-1-yl)-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}propanamide
{[5-(oxolan-2-yl)thiophen-2-yl]methyl}(propyl)(pyridin-3-ylmethyl)amine
N-benzyl-N-methyl-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
2-chloro-4-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenol
N-[2-(4-chlorobenzenesulfonamido)ethyl]-3-(pyridin-4-yl)propanamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(methoxymethyl)piperidine
2-(cyclopentylmethyl)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[1-(4-chlorophenyl)cyclobutyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[(4-ethylphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-[(1R,2R)-2-(benzyloxy)cyclohexyl]-5-methyl-1,3,4-oxadiazol-2-amine
3-[(1-acetylpiperidin-4-yl)oxy]-N-(2-hydroxy-2-phenylethyl)-4-methoxy-N-methylbenzamide
ethyl 2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylate
1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}piperidine-2-carboxylic acid
N-(1-methyl-1H-1,2,4-triazol-3-yl)-3-(propoxymethyl)pyrrolidine-1-carboxamide
4-(3-fluorophenyl)-3-(1H-indol-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-methoxyethyl)-5-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
N-ethyl-3-(3-fluorophenyl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide