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3-(1H-1,3-benzodiazol-1-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-cyclohexyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
ethyl 1-[2-(dimethylamino)ethyl]-5-[(4-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)prop-2-ene-1-sulfonamide
3-(2,3-dichlorophenyl)-6-methoxypyridazine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
N-methyl-3-{[2-(4-methylpentyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
[5-(2-ethylphenyl)-1H-1,3-benzodiazol-2-yl]methanol
N-[(2S,4R,6S)-2-benzyl-6-(1-methyl-1H-1,2,3-benzotriazol-5-yl)oxan-4-yl]acetamide
N,N-diethyl-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
2-(3-chloro-4-hydroxyphenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]acetamide
8-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
3-[4-(2-oxopyrrolidin-1-yl)phenyl]-1-[3-(pyridin-3-yl)propyl]urea
(1R,5R)-3-(2-methylpyrimidine-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)quinolin-8-ol
2-[(2S)-2-(methylamino)propanoyl]-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-(4-chloro-2-methylbenzoyl)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
[(2S,6S)-4-(5-chloro-2-methoxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-{[5-(3-acetylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-N-methylacetamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
[(3R,4R)-1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-4-yl)pyridine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1H-pyrrole-3-carboxamide
2-cyclohexyl-1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-hydroxy-4-methylpentan-1-one
N-ethyl-2-oxo-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxaspiro[4.4]nonane-4-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N,2-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]furan-3-carboxamide
methyl 3-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}benzoate
5-[1-(3,5-dimethylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrazin-2-ol
ethyl 4-[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]piperidine-1-carboxylate
3-phenyl-N-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]propanamide
(1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
6-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
2-[2-(3-propoxypiperidin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-ol
2-{1-[1-(furan-2-yl)ethyl]-1H-imidazol-2-yl}-1-(4-methoxyphenyl)-1H-imidazole
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-4-phenoxybutan-1-one
1-(diphenylmethyl)-4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-1,2,3-triazole
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
9-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
3-(3-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}benzamide
1-{4-[(cyclohexylmethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-(4-fluorophenyl)-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]morpholine