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N-{2-[ethyl(methyl)amino]-2-methylpropyl}-6-(propan-2-yl)pyrimidin-4-amine
5-{[(1-hydroxycyclohexyl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[(3S)-3-phenylbutanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2-chloro-4-fluorophenyl)methyl]-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
3-(2-methoxyethyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylic acid
5-methoxy-N-methyl-4-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-4H-pyran-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)-2-(3-fluorophenyl)-N-methylacetamide
1-[2-(difluoromethoxy)benzoyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-{3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]benzenesulfonyl}azetidin-3-ol
9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}but-2-ynamide
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-acetamidoethyl)piperidine-3,5-dicarboxamide
1-(4-{[(2R,5S)-5-(2H-1,3-benzodioxol-5-ylmethyl)oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
2-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)ethan-1-ol
6-phenyl-3-[4-(piperidin-1-yl)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)pyridine
1-(4-methoxyphenyl)-5-methyl-4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
3-{1-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propyl]piperidin-2-yl}pyridine
5-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
1-ethyl-4-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
3-(benzyloxy)-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-methoxyethyl)-N,5-dimethyl-1H-pyrazole-4-carboxamide
3-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-ethyl-1-(oxan-4-ylmethyl)urea
2-(3-fluorophenoxymethyl)-N-[(1-methylpiperidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-[3-oxo-9-(pyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
4-[(4-fluorophenyl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
N5-cyclooctyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
N-[(2-fluorophenyl)methyl]-3-[1-(pyridine-3-carbonyl)piperidin-3-yl]propanamide
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
(1S,5R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-chloro-1H-pyrazole-3-carbonyl)-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(2-methylphenyl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
1,3-dimethyl-6-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1H-imidazole-4-carboxylate
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]benzamide
3-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-cyclopentyl-4-methoxybenzamide
3-{[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3,4-dimethoxyphenyl)methyl]-2-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)acetamide
N-(2,2-difluoroethyl)-4-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
1-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-dihydroquinoxalin-2-one
3-({1-[4-(piperidin-1-ylmethyl)benzoyl]piperidin-4-yl}oxy)pyridine
1-({2-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carbonitrile
2-(5-acetylthiophen-3-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
N-[3-(4-ethoxyphenyl)propyl]-2-(morpholin-3-yl)acetamide
1-methyl-2-({3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-imidazole