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N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]pyridazin-3-amine
N3-[3-(2-fluorophenyl)propyl]piperidine-1,3-dicarboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
6-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-ethyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-6-oxopiperidine-3-carboxamide
5-methyl-N4-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyrimidine-2,4-diamine
(6-methylhept-5-en-2-yl)[3-(pyridin-2-yl)propyl]amine
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(quinolin-5-ylmethyl)piperidin-3-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(3S,4S)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-{2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-chloro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
8-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]methyl}-1-(2-methoxyethyl)-6-methyl-1,2-dihydroquinolin-2-one
1-[2-(morpholin-4-yl)-2-oxoethyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2-methylpropyl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2-oxazole-5-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-[(3-methoxyphenyl)methyl]piperidin-2-one
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-(2-methylpropyl)morpholine
2-{4-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]pyrimidin-5-yl}acetic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-ethylpiperazine
4'-(3-fluoropropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-ethyl-4-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-2-one
(4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-3,3,4-trimethylpiperidin-4-ol
3-fluoro-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}benzamide
3-[3-(furan-2-yl)-1H-pyrazol-1-yl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-{4-[(1-ethyl-1H-indol-4-yl)methyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(pyrrolidine-1-sulfonyl)piperazine
5-(3-acetylphenoxymethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-pyrazole-3-carboxamide
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N,1-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-2-carboxamide
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-[(4-fluorophenyl)methyl]-2-(1-methylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}-4,4-difluoropiperidine
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(thian-4-yl)piperazine
2-(1,2-benzoxazol-3-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-[3-(4-hydroxyphenyl)propanoyl]piperazin-2-one
methyl (2S,4R)-4-(dimethylamino)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidine-2-carboxylate
(3S,4S)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-2-(1H-pyrazol-1-yl)acetamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzoxepine-4-carboxamide
N-(4-fluoro-2-methylphenyl)-2-{[1-(4-methylpiperazin-1-yl)propan-2-yl]amino}acetamide
5-methyl-4-[(oxolan-3-yl)amino]-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
8-[4-(1H-indol-3-yl)butan-2-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (1R,3S,3aR,6aS)-1-benzyl-3-(furan-3-yl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2,1-benzoxazole-3-carboxamide