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ethyl 4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-(furan-2-ylmethyl)-5-{1-[2-(pyridin-2-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-amino-6-[3-fluoro-5-(trifluoromethyl)phenyl]-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-methyl-4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-7-methyl-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
6-[2-(2-methylpropoxy)phenyl]pyridine-2-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-3-yl]propan-1-ol
5,5-dimethyl-3-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,3-oxazolidine-2,4-dione
1-cyclopentanecarbonyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
2-methyl-3-(1,4-oxazepane-4-carbonyl)-N-(pyridin-2-ylmethyl)aniline
1-(4-methylpiperazin-1-yl)-3-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)propan-2-ol
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3,4-dimethoxyphenyl)methyl]-N-phenylpiperidin-3-amine
4-(2-methyloxolane-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-(1-ethylpiperidin-4-yl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}acetamide
N-benzyl-5-methoxy-N-(1,3-thiazol-2-ylmethyl)-1H-indole-2-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(2,3-dimethylphenyl)-N'-{2-[(2-ethylphenyl)carbamoyl]ethyl}propanediamide
N-[2-(6-methylpyridin-2-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(thiophen-2-yl)azetidin-1-yl]propan-1-one
N-(2-methyl-1-benzofuran-7-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-[4-({1-[(4-fluorophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)piperazin-1-yl]propan-1-one
3-[5-({[1-(4-methylphenyl)ethyl]carbamoyl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-benzyl-6-hydroxy-1,4-diazepane-1-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
1-(4-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
1-(1-methyl-1H-pyrrol-2-yl)-2-[2-(pyridin-2-yl)piperidin-1-yl]ethane-1,2-dione
2-{[(5-{1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
1-[1-(1-ethylpiperidine-4-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
methyl 4-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-4-oxobutanoate
2-(4-hydroxyphenyl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)but-3-enamide
N3-cyclooctyl-N5-[2-(methylsulfanyl)ethyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-acetyl-3-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
3-cyano-N-{[1-(cyclohex-2-en-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}benzamide
(2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-[(1H-1,2,4-triazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(4-methoxyphenyl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
ethyl 4-(3-{[2-(4-methoxyphenyl)acetamido]methyl}piperidin-1-yl)piperidine-1-carboxylate
1-[(5-methylthiophen-2-yl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-phenyl-1,2-oxazole-3-carboxamide
methyl 2-{1-[(2,5-dimethoxyphenyl)carbamoyl]pyrrolidin-3-yl}acetate
2-cyclopropyl-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)-2,6-dimethoxyphenol
[(3R,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-[(2-fluorophenyl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
6-(methoxymethyl)-2-(4-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one