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1-[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]azepane
2-[(2,6-dichlorophenyl)methyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N,2,6-trimethylpyrimidine-4-carboxamide
1-{2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}ethan-1-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-2-propyl-1,3-thiazole-4-carboxamide
(1S,5R)-3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-[1-(1-cyclobutylpiperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
1-{6-chloro-3-[(3,4-dimethylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}azocane
4-{1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
2-methyl-N-{1-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-hydroxy-4-methyl-N-[3-(pyridin-3-yl)propyl]pentanamide
methyl 2-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})carbamoyl]piperidine-1-carboxylate
ethyl 1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-4-carboxylate
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-(2-{[3-(4-fluorophenyl)-1H-pyrazol-5-yl]formamido}ethyl)piperidine-3-carboxamide
2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
N-[3-(3-fluorophenyl)phenyl]-1-(3-hydroxy-2,2-dimethylpropyl)piperidine-4-carboxamide
N-[2-(4-ethoxyphenyl)phenyl]-2-methoxyacetamide
2-cyclopropanecarbonyl-8-(5-fluoropyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-(8-methoxyquinolin-5-yl)-N,N-dimethylpyridazin-3-amine
3-{3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}pyridine
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(4-methoxyphenyl)-2-methylpiperazine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
2-{4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-1-yl}-1,3-benzothiazole
(3R,4S)-4-cyclopropyl-1-[1-(2-fluorophenyl)piperidin-4-yl]pyrrolidin-3-amine
2-({[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}amino)-2-methylpropan-1-ol
(1S,6R)-9-{2-[(4-hydroxyquinazolin-2-yl)sulfanyl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-ethyl-N-(oxan-4-ylmethyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
7-[2-(2-chloro-4-fluorophenoxy)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(azepane-1-sulfonyl)-5-{pyrazolo[1,5-a]pyridin-7-yl}benzoic acid
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
N-[3-(2-ethoxyphenyl)propyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
methyl 4-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)benzoate
2-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
N-[3-(2-methoxyphenyl)propyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-7-methanesulfonyl-4-methylquinazoline
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenylethan-1-one
(3S,4R)-4-phenyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidine-3-carboxylic acid
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-cyclopentyl-2-({[5-fluoro-2-(trifluoromethyl)phenyl]methyl}amino)propanamide
1-(6-hydroxy-4-{2-[(4-methylphenyl)methyl]benzoyl}-1,4-diazepan-1-yl)ethan-1-one
2-ethyl-N-(3-phenylcyclobutyl)-2H-1,2,3,4-tetrazol-5-amine
4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-2-propylpyridine
dimethyl[(4-{1-[(3-methylpyridin-2-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
(2S)-1-methyl-N-[3-(3-phenylpropanamido)phenyl]pyrrolidine-2-carboxamide
(2-methoxyethyl)({[2-(5-methylfuran-2-yl)phenyl]methyl})(oxolan-2-ylmethyl)amine