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5-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-3-methylquinoxaline
2-({[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
1-[3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N3-cyclohexyl-1-(2-methylpropyl)-N5-[2-(methylsulfanyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,9aR)-1-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
[2-(2,3-dimethylphenoxy)ethyl](methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)-1-azabicyclo[2.2.2]octane
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]thiophene-2-carboxamide
N-ethyl-2-methyl-3-[(pyridin-3-ylmethyl)amino]-N-(pyridin-4-ylmethyl)benzamide
4-methyl-N-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-1,2,3,6-tetrahydropyridine-1-carboxamide
methyl N-{2-[(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}carbamate
N-[3-(cyclohexylsulfanyl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-ethoxy-2-hydroxypropyl)benzamide
N-ethyl-5-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(2,3,6-trifluorophenyl)acetamide
4-fluoro-2-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}phenol
3-{4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)pyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3,5-dimethylbenzamide
N-(1,3-benzothiazol-2-ylmethyl)-2-(ethylamino)-N,4-dimethyl-1,3-thiazole-5-carboxamide
3-{5-[1-(3-chlorophenoxy)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
1-{[1-(2-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methoxy-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
3-[(3R,4S)-1-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-(2-{1-[3-(3-methoxy-4-methylphenyl)propanoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-{1-cyclohexyl-5-[1-(4-methoxyphenyl)cyclopropyl]-1H-1,2,4-triazol-3-yl}acetamide
7-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-benzyl-8-(cyclohex-3-en-1-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
5-benzyl-N-[1-(hydroxymethyl)cyclopentyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-fluoro-6-[(1E)-pent-1-en-1-yl]benzamide
4-(5-methylpyridin-2-yl)-1-[(E)-2-phenylethenesulfonyl]piperidin-4-ol
ethyl 4-[2-(1H-pyrazol-1-yl)butanoyl]piperazine-1-carboxylate
7-[(2,3-difluorophenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-chlorophenyl)-5-(propane-1-sulfonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
(3R,4R)-4-amino-1-({2-[(4-chlorophenyl)methoxy]phenyl}methyl)piperidin-3-ol
3-(4-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
3-[4-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
4-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-imidazol-2-one
2-(2,6-dimethoxy-4-methylphenyl)-2-[(2-hydroxyethyl)(methyl)amino]acetic acid
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(propan-2-ylsulfanyl)acetamide
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[1-(thiophen-2-yl)propyl]-1H-pyrazole-3-carboxamide
dimethyl[3-(2-{1-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
3-(propan-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-oxazole-5-carboxamide
(1S,5R)-3-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[2-(cyclopropylmethyl)-4-{[3-(methylsulfanyl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one