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9-[(2,4-difluorophenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-cyclopentyl-N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-cyclopentyl-4-[8-(trifluoromethyl)quinolin-4-yl]piperazin-2-yl}ethan-1-ol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
N-methyl-2-[N-(3-methylphenyl)methanesulfonamido]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
4-[(1S,2S)-2-hydroxycyclohexyl]-N-[4-(methylsulfanyl)phenyl]piperazine-1-carboxamide
3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-6-(pyridin-4-yl)-1,2-dihydropyridin-2-one
(3aR,6aR)-2-(2-methoxyethyl)-5-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-3-fluoro-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}benzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
1-{1-[(2-fluoro-3-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-({1-[6-(thiophen-3-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-ethyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,4S)-2-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane
1-ethyl-5-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
1-(2,3-dihydro-1H-inden-2-yl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[1-(2-methylpropyl)cyclopropyl]amino}methyl)piperidin-2-one
N-[(4-phenyloxan-4-yl)methyl]-6-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(pyrimidin-2-yl)piperidin-3-amine
3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5,6,7,8-tetrahydroquinoline
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperazine
N-{2-[2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamido]-4-methylphenyl}benzamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-1,3-benzodiazole-6-carboxylic acid
3-(2-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-tert-butyl-4-hydroxy-N-(2,2,2-trifluoroethyl)pyrimidine-5-carboxamide
2-(5-{1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
5-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
1-methyl-4-{1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
4-({4-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]piperazin-1-yl}methyl)-2-methylphenol
3-(4-hydroxyphenyl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-hydroxy-3-({[(1-hydroxycyclohexyl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
1-(methoxymethyl)-N-[(3R,4S)-1-methyl-4-phenylpyrrolidin-3-yl]cyclobutane-1-carboxamide
2-(3-hydroxyphenyl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
5-methoxy-1-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-indole-2-carboxamide
N-cyclopentyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
6-(aminomethyl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]pyrimidin-4-amine
N'-(adamantan-1-yl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanediamide
1-[5,6,7-trimethoxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
2-(2-phenylethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
1-({4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-1,2,3,4-tetrazole
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid