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2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoacetamide
3,5-dimethyl-6-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
N-[(3R,4S)-1-(2,5-dimethylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-1-yl}phenol
2-(pyridin-2-ylsulfanyl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
1-{3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}propan-1-one
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-4-fluorobenzamide
8-(2-ethoxyethyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(2S)-4-methanesulfonyl-2-[(2-propyl-1,3-thiazol-4-yl)formamido]butanoic acid
1-[(1s,4s)-4-aminocyclohexyl]-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
11-{[(2,6-difluorophenyl)methyl]amino}-4-[3-(pyridin-4-yl)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-tert-butyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-5-oxopyrrolidine-3-carboxamide
N-(9H-fluoren-9-yl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl](oxolan-2-ylmethyl)amine
2-{4-[(1-methyl-1H-indol-5-yl)methyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
N-[(4-chlorophenyl)methyl]-4-(dimethylamino)azepane-1-carboxamide
[(3S,5R)-1-(2-methoxypyridine-4-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
4-{3-cyclobutyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-N-methylbenzene-1-sulfonamide
4-[6-(dimethylamino)pyrazin-2-yl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
(2S,4R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-hydroxypyrrolidine-2-carboxylic acid
5-({[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
2-methyl-8-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{[2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
2-methyl-3-{[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}quinoxaline
ethyl 4-[3-(2-hydroxyphenyl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
N-[(1S,2R)-2-aminocyclobutyl]-2-(benzyloxy)acetamide
(3R,4R)-1-[(4-methoxypyridin-2-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-[2-(1,3-benzothiazol-2-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 6-(2-cyclopropylacetyl)-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclopentyl-4-({methyl[(2E)-2-methylbut-2-en-1-yl]amino}methyl)pyrrolidin-2-one
1-(2-methoxyacetyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-3-carboxamide
2-[2-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]urea
8-{[(4-chlorophenyl)methyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3aS,6aS)-2-{[2-(benzyloxy)phenyl]methyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylate
3-{1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-(1-{[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
4-(5-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
N-ethyl-5-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyrimidin-2-amine
(2S,4S)-1-benzyl-4-{[(4-chlorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-fluorophenyl)-2-hydroxyethan-1-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dipropylacetamide
N-[(3R,4S)-1-(1,3-dihydroxypropan-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(4-methylphenoxy)acetamide
3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide