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1-(pyridin-2-yl)-4-[(3-{[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
(1S,5R)-3-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aS)-1-methyl-5-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-octahydropyrrolo[3,4-b]pyrrole
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-methylpropyl)piperidine-3,5-dicarboxamide
methyl 5-(5-methoxy-1H-indole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[3-(trifluoromethyl)-1H-pyrazol-5-yl]methyl}amine
2-{[4-(4-methylphenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-ethyl-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 2-{[2-(dimethylamino)ethyl]carbamoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
N-[(3R,4R)-3-hydroxy-1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-4-yl]pyridine-2-carboxamide
5-methanesulfonyl-N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethylpyrimidin-4-amine
1-{4-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-oxobutyl}pyrrolidin-2-one
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(2-oxopyrrolidin-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
ethyl[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](oxan-2-ylmethyl)amine
1-[4-(3-methoxyphenyl)phenyl]-N-(1-methoxypropan-2-yl)piperidin-4-amine
1-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
5-(3-fluorophenyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1,2,4-triazin-3-amine
2-(4-chlorophenyl)-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]morpholine
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
1-(dimethyl-1,3-oxazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-2-methoxybenzoic acid
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,8-dimethylquinoline
(2R,3R)-3-({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(3-fluorophenyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
3-[1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)piperidin-3-yl]propanamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,6-dihydroxypyridine-3-carboxamide
2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
N-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-(cyclopropylmethyl)-1-(3-methoxypropyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(1R,2S)-N-butyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]cyclohexane-1-carboxamide
(2R,6S)-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,6-dimethylmorpholine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(pyridin-4-yl)ethyl]benzamide
2-[(3-{[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
N-[4-(1H-imidazol-1-yl)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
6-ethyl-5-methyl-N4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrimidine-2,4-diamine
1-[(3,4-dimethylphenyl)methyl]-4-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperazin-2-one
7-(1-benzothiophen-3-yl)-4-(3,5-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,7aS)-1-ethyl-4-(9H-fluorene-9-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{5-[2-(benzenesulfonyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[4-(3-methylphenyl)phenoxy]propanamide
3-[1-(morpholine-4-sulfonyl)piperidin-3-yl]benzoic acid
2-[3-oxo-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
N-butyl-N-methyl-3-(1,4-oxazepan-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-methoxy-5-{1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}benzoic acid
2-(methylamino)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyridine-3-carboxamide
4-{[(quinolin-2-yl)amino]methyl}-1λ6-thiane-1,1-dione
5-phenyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(2-chloropyridin-3-yl)methyl]methylamine