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2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-(3-methoxyphenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrazole-4-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]furan-2-carboxamide
4-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4H-1,2,4-triazole
6-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)-9H-purine
methyl 4-{[3-(3-chlorophenyl)phenyl]carbamoyl}piperidine-1-carboxylate
1-(4-fluorophenyl)-4-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)butane-1,4-dione
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
3-{2-[(dimethylamino)methyl]phenyl}-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
6-(furan-2-ylmethyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
4-[6-(2,4-dimethoxyphenyl)pyridazin-3-yl]thiomorpholine
2-methyl-N-[(2-phenoxypyridin-3-yl)methyl]-1,8-naphthyridine-3-carboxamide
7-(cyclobutylmethyl)-2-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[3-(2-methylphenoxy)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
5-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-3-phenyl-1,2,4-oxadiazole
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-(2-phenoxyethyl)piperazine
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-ethoxyethan-1-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(1H-imidazol-2-yl)benzamide
5-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-(2,5-difluorophenyl)-4-(pyrrolidine-1-sulfonyl)piperazine-1-carboxamide
(3E)-N-[2-(2-phenoxyethoxy)phenyl]pent-3-enamide
1-[2-(morpholin-3-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(ethylamino)pyrimidine-5-carboxamide
methyl 2-[4-(2-phenoxyethyl)piperazine-1-carbonyl]piperidine-1-carboxylate
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl]propanoate
N-[(2-chloro-6-fluorophenyl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-{5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
N-({1-[4-(thiophen-2-yl)butanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
3-{[(3S)-3-(dimethylamino)azepan-1-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
3-(pentan-2-yl)-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[4-(4-methoxybutyl)piperazine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
8-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
(5S,9aS,9bS)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-phenyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
ethyl 1-[(3-acetylphenyl)methyl]-4-benzylpiperidine-4-carboxylate
3-phenyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
methyl 7-oxo-3-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{5-[5-(4-methoxyphenyl)furan-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
3-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}quinolin-7-ol
2-(2,2-dimethyloxan-4-yl)-1-[2-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
benzyl(methyl)[(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]amine
1-({1-[(benzyloxy)carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-methyl-N-(2-phenylpropyl)-3-propyl-1H-pyrazole-5-carboxamide