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2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-fluorophenyl)pyrimidine
N-benzyl-N-methyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-3-amine
ethyl 1-(5-acetylthiophene-2-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]pyridine-2-carbonitrile
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)-1H-pyrazole
naphthalen-1-yl (7R,9aR)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-(4-chloro-2-ethylphenyl)-2-(hydroxymethyl)azepane-1-carboxamide
7-(cyclopropylmethyl)-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decane
4,5-dimethyl-6-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidine
(3R,4R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(pyridin-3-yl)propanamide
1-methyl-N-[3-(morpholin-4-yl)propyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-{2-[3-cyclopentyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
2-[7-(hydroxymethyl)-9-(3-methoxypropanoyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
4-(cyclopropylmethyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-{3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]phenoxy}acetamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
6-(2-aminoethyl)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethylpyrimidin-4-amine
3-benzyl-4-[2-(1H-imidazol-2-yl)benzoyl]piperazin-2-one
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
4-(3-ethylpiperazin-1-yl)-N-(2-fluoro-5-methylphenyl)-4-oxobutanamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
6-methoxy-4-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
3-(5-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
4-(2-chloro-5-methylphenyl)-6-(methoxymethyl)pyrimidine
3-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-7,8-dimethyl-3,4-dihydroquinazolin-4-one
N-{5-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,3-thiazol-2-yl}acetamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
2-{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-oxoethoxy}acetamide
1-(2-ethoxyethyl)-N-[(4-methylphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropan-1-amine
5-[2-(butan-2-yloxy)phenyl]-1-propyl-1H,4H-pyrazolo[3,4-d]imidazole
(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
dimethyl(2-{2-[1-(naphthalene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
1-[4-(cyclobutylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-[1-(3-methoxy-4-methylbenzoyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(4aS,8aR)-1-(2-aminoethyl)-N-[(3-fluorophenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
2-[2-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)phenoxy]acetic acid
N-[1-(hydroxymethyl)cyclopentyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
9-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(2-phenylpropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
5-{1-[2-(3,5-difluorophenyl)-1H-imidazol-1-yl]ethyl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-ethyl-5-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}pyrimidine
(3S,4R)-3-benzyl-4-methyl-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-(1-{2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propan-2-yl)piperazine
N-[2-methyl-3-(methylcarbamoyl)phenyl]-4-(thian-4-yl)piperazine-1-carboxamide