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1-{1-[6-(2,4-difluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-{4-[methyl(2-phenoxyethyl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
5-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
[3-(hydroxymethyl)-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)benzamide
5-[3-(methoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
4-(2,6-dimethylpyridin-3-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidin-2-amine
1-cyclohexyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[4-(2,3-dihydro-1H-inden-2-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-cyclopropyl-5-{thieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(3-methyl-1,2-benzoxazol-5-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,4R)-1-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
N-cyclohexyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-fluoro-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-2-carboxamide
N,N-dimethyl-2-(4-methylpentyl)morpholine-4-sulfonamide
N-benzyl-6-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
N-(1,2-oxazol-5-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
1-[(5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}furan-2-yl)methyl]pyrrolidine
1-[2-methoxy-6-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-({[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]oxy}methyl)pyridine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}-1,4-diazepan-5-one
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
N-[2-(1H-indol-1-yl)ethyl]-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-methyl-N-{3-oxo-3-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)oxolane-3-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
3-(quinolin-6-ylmethyl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
1-[(1-hydroxycyclohexyl)methyl]-3-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-[2-(diethylamino)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-ethyl-N-[2-methyl-5-(3-methyl-1H-1,2,4-triazol-5-yl)phenyl]butanamide
8-methoxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-{2-[3-(2-methylphenyl)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}butanamide
(1R,5S,6S)-6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
4-[(4-ethylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(6-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-yl)morpholine
1-[1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
benzyl N-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl}carbamate
1-{[(3R,4R)-1-(6-ethyl-2-methylpyrimidin-4-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-ethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-[2-(3-propanamidophenoxy)acetyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(2-hydroxy-5-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
({1-[1-(2-ethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
5-hydroxy-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)pyrazine-2-carboxamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aR)-2-(5-chlorothiophene-2-carbonyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid