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5-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(propylcarbamoyl)pyrrolidine-2-carboxylic acid
2-cyclobutyl-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-6-methylpyridin-3-ol
6,6-dimethyl-1-phenyl-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-(4-fluorophenyl)-1-(1H-imidazol-4-ylmethyl)piperidin-3-amine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(3-hydroxypropanoyl)piperidine-4-carboxamide
(1R,9S)-5-amino-3-(4-chloro-1-methyl-1H-indazol-3-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-(2-methoxyethyl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-(propan-2-yloxy)benzamide
1-(2-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-(adamantan-1-yl)-N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}acetamide
5-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
1-{1-[1-(1,4-dimethylpiperidine-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
3-(4-fluorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]cyclopentanecarboxamide
4-[(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-(azocan-1-yl)-N-{2-[(2-methoxyphenyl)carbamoyl]ethyl}propanamide
2-fluoro-N-{3-[3-(2-methylphenoxy)azetidin-1-yl]-3-oxopropyl}benzamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
(1-methyl-1H-imidazol-2-yl)({1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl})methanol
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(methoxymethyl)piperidine
1-[4-(3-hydroxyphenyl)piperidin-1-yl]-2-(1-methylpyrrolidin-2-yl)ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(7-methoxy-4-methyl-2-oxo-2H-chromen-3-yl)acetamide
2-(4-fluoro-2-methoxyphenyl)-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)acetic acid
N-(1-{7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
5-(hydroxymethyl)-2-methyl-4-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-3-ol
N-cyclopentyl-3-[5-(oxan-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
4-ethanesulfonamido-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
2-(2-chloro-4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)acetamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-methyl-1H-indazol-5-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(3-phenylpyrrolidin-1-yl)acetamide
3-methyl-4-({3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
2-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethan-1-ol
ethyl 1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
3-({4-[1-(prop-2-ene-1-sulfonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-({1-[3-(2-oxoimidazolidin-1-yl)benzoyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
2-(4-methanesulfonylphenyl)-6,7-dimethoxyquinazolin-4-amine
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
5-[(2R)-2-methylpiperazine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
2-(4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
[(3-fluorophenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine