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(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(pyridin-2-ylmethyl)-decahydro-2,7-naphthyridine-2-carboxamide
1-cyclopentyl-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
3-(piperazine-1-sulfonyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
4-[2-(methylsulfanyl)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[(3R,4S)-4-cyclopropyl-1-(5-methyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
2-(4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}morpholin-3-yl)acetic acid
(1S,5R)-3-(3,4-difluorobenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(benzyloxy)-5-[3-(methoxymethyl)-1H-1,2,4-triazol-5-yl]pyridine
2-methyl-4-(4-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
2-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-(cyclohexylmethyl)-N-cyclopropyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
5-cyclobutanecarbonyl-1'-(furan-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
methyl 3-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}sulfonyl)thiophene-2-carboxylate
6-methyl-2-{2-[(propan-2-yl)carbamoyl]phenyl}pyridine-3-carboxamide
1-(3-chlorophenyl)-4-(7-methyl-1-benzofuran-2-carbonyl)piperazin-2-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methyl-N-(2-phenylethyl)acetamide
(3S,5R)-1-benzyl-N3-butyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
N'-(3-ethylphenyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]butanediamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-{3-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]propyl}-4-methylbenzene-1-sulfonamide
(3S,4R)-1-cyclohexanecarbonyl-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-(2,3-dihydro-1H-inden-1-yl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-phenoxy-N-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-[1-(2,6-difluoro-3-methylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-{[3-methyl-7-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(cyclopropylmethyl)-5-(3-fluorophenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
1-{1-[(5-chlorothiophen-2-yl)methyl]azetidin-3-yl}-2-methylpiperidine
N-(furan-2-ylmethyl)-6-methyl-4-oxo-N-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3-methoxyphenyl)propanamide
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-oxo-1-(prop-2-en-1-yl)piperidine-3-carboxamide
3-{[(1-cycloheptyl-5-oxopyrrolidin-3-yl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
1-[2-(8-methoxy-2-methylquinolin-5-yl)pyrimidin-4-yl]piperidin-4-ol
N'-(2,5-dimethylphenyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]propanediamide
4-{5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]furan-2-carbonyl}morpholine
(1S,5R)-6-(2-methylbenzenesulfonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-chloro-2-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
2-(4-fluorophenyl)-N-(piperidin-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
8-(pyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
dimethyl({2-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl})amine
1-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}azepan-4-amine
4-[(6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]morpholine
9-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-{2-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
(1R,9aR)-1-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-octahydro-1H-quinolizin-1-ol
2-amino-4-(2,6-dichloro-3-hydroxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile